LGD -4033 (Ligand Yob) 10mg 100 Ntseg Cov Lus Qhia Tshwj Xeeb*
Kws muag tshuaj -} qib raw cov ntaub ntawv|LGD-4033 (Xaiv Androgen Revenor Modulator)
Tshuaj lom neeg npe: 4 - ((R) -2 - ((R) -2,2,2-devrluoro-1-hydrolidin-1-YL) -2- (Trifluoromethyl) Benzonitrile
Tus lej: 1165910-22-4
Einecs tooj: Kom raug muab
Cov Qauv Molecular: C₁₄h₁₂f₆n₂o
Molecular hnyav: 338.25
Melting taw tes: 158-160 degree
Zog: Dawb Crystalline Hmoov
Purity: ntau dua los yog sib npaug rau 98% (HPLC sim)
Cov khoom tseem ceeb
LGD-4033 yog aKev xaiv siab Androgen Revenor Modulator (SARM) uasyog siv dav hauvKev loj hlob ntawm cov leeg, cov osteoporosis kev tshawb fawb, thiab tshuaj kis lasVim nwsmuaj lub zog anabolic kev ua si thiab cov kev mob tshwm sim qis.
✅ Precise Targing Mechan:
Siab receptor affinity: High affinity rau androgen receptor (Ki=~ 1nm)
Nqaij Nqaij Xaiv: Cov ntaub ntawv ua yeeb yam tag nrho hauv cov leeg thiab cov pob txha
Prostate kev nyab xeeb: Cuam tshuam kev ua si hauv cov nqaij mos
✅ Zoo heev Anabolic:
Nce cov nqaij ntshiv lub cev loj: Cov kev tshawb fawb soj ntsuam tau pom tias muaj qhov qhib - Nyob rau hauv cov nqaij ntshiv lub cev
Lub Zog Li: Txhim kho cov leeg nqaij thiab lub zog thiab kev ua kis las
Pob Txha Kev Noj Qab Haus Huv: Nce pob txha ceev thiab txhim kho pob txha ua tau zoo
✅ Cov yam ntxwv nyab xeeb:
Hypoandrogenicity: Tsawg Txiaj Fwv ntawm Androgenic phiv
Tsis muaj kev sib cav: Tsis muaj hloov dua siab tshiab rau estrogen, tsis muaj kev pheej hmoo ntawm dej rov qab
Tsawg Hepatotoxicity: Zoo zam los ntawm daim siab ntawm kho cov koob tshuaj
Cov kev siv raws tu qauv
1. Kev Tshawb Fawb Txog Kev Tshawb Fawb:
Pib koob tshuaj:
1 mg ib zaug txhua hnub
Kev Ntsuam Xyuas Kev Ntsuas Rau 1 Lub Limtiam
Escalating koob tshuaj:
Lim tiam 2: 2 mg / hnub
Los ntawm 3 lub lim tiam dhau los: kho rau 3-5 mg / hnub raws li kev kawm xav tau
Koob tshuaj ntau tshaj plaws:
Qhov kev kawm dose tsis tshaj 10 mg / hnub
2. Siv kev voj voog:
Luv - lus kawm: 4-6 lub lis piam
Ntev - lub sij hawm kawm: 8-12 lub lis piam (yuav tsum muaj kev soj ntsuam ze)
Tshaj tawm - kev mus kuaj xyuas: Txuas ntxiv saib xyuas 4 lub lis piam tom qab siv tshuaj noj
3. Saib xyuas cov ntsuas:
Cov hauj lwm ua hauj lwm zoo:
Hloov pauv ntawm cov nqaij ntshiv lub cev
Cov leeg ua kom muaj zog kuaj
Kev Ntsuas Pob Txom
Qhov ntsuas kev nyab xeeb:
Daim Siab Ua Haujlwm Kev Ntsuam Xyuas
Cov qib ntshav lipid
Hormone Qib Kev Ntsuam Xyuas
Vim li cas thiaj xaiv LGD-4033 cov khoom siv raw?
Siab Xaiv: Muaj kev xaiv thiab muaj kev sib cav heev rau Androgen Receptors
Cov leeg muaj zog: Cov kev tshawb fawb soj ntsuam tau ua pov thawj qhov tseem ceeb nce nyob rau hauv cov nqaij ntshiv lub cev thiab cov leeg kom muaj zog
Kev tshawb nrhiav tus nqi: Nws muaj cov tseem ceeb tshawb fawb hauv kev kho mob ntawm cov leeg leeg atrophy thiab osteoporosis
Lub ntsiab
LGD-4033 yogIb qho cuab yeej tseem ceeb hauv kev tshawb fawb ntawm kev xaiv cov androgen receptor modulators.DhauKev tshawb fawb txuj ci txheej txheem,Nws tuaj yeem tsim rau hauvNtau cov ntaub ntawv muab tshuaj, suav nrog cov ntsiav tshuaj ntawm qhov ncaujCov. Xaiv peb kom ntseeg tausiab -} Purity raw cov ntaub ntawv, kev txhawb nqa kev ua haujlwm, thiab muaj txhij txhua {{1} kev pab muag khoom.
Xav taudab tsi, thov hu raupeb
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Ntawv xov |
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Cim npe nrov: LGD 4033 10 mg * 100 / lub raj mis Stromusc slomsets ntawm qhov rooj ntawm qhov ncauj ntawm daim ntsiav tshuaj ntawm qhov ncauj ntawm daim ntsiav tshuaj ntawm daim ntsiav tshuaj

