LGD 4033 10 ml * 100 / lub raj mis Stromusc slarusc sarmsts

LGD 4033 10 ml * 100 / lub raj mis Stromusc slarusc sarmsts
Khoom Taw qhia:
LGD4033 yog qhov muaj zog sarm40 tau nce siab heev ntshiv lub cev thiab pob txha ceev los ntawm kev sib tw thiab cov pob txha, nrog zoo tsis muaj cov kev mob thiab cov kab mob. Cov kev tshawb fawb soj ntsuam tab tom pib rau kev kho mob ntawm cov dystrophy thiab txha osteoporosis. Nws yog qhov tsim txiaj (5-10 mg / hnub) thiab muaj kev tshawb nrhiav tus nqi rau kev ua kom raug mob thiab txhim kho lub cev kev txhim kho.
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Kev tsis

LGD -4033 (Ligand Yob) 10mg 100 Ntseg Cov Lus Qhia Tshwj Xeeb*

Kws muag tshuaj -} qib raw cov ntaub ntawv|LGD-4033 (Xaiv Androgen Revenor Modulator)

Tshuaj lom neeg npe: 4 - ((R) -2 - ((R) -2,2,2-devrluoro-1-hydrolidin-1-YL) -2- (Trifluoromethyl) Benzonitrile

Tus lej: 1165910-22-4

Einecs tooj: Kom raug muab

Cov Qauv Molecular: C₁₄h₁₂f₆n₂o

Molecular hnyav: 338.25

Melting taw tes: 158-160 degree

Zog: Dawb Crystalline Hmoov

Purity: ntau dua los yog sib npaug rau 98% (HPLC sim)


Cov khoom tseem ceeb

LGD-4033 yog aKev xaiv siab Androgen Revenor Modulator (SARM) uasyog siv dav hauvKev loj hlob ntawm cov leeg, cov osteoporosis kev tshawb fawb, thiab tshuaj kis lasVim nwsmuaj lub zog anabolic kev ua si thiab cov kev mob tshwm sim qis.

Precise Targing Mechan:

Siab receptor affinity: High affinity rau androgen receptor (Ki=~ 1nm)

Nqaij Nqaij Xaiv: Cov ntaub ntawv ua yeeb yam tag nrho hauv cov leeg thiab cov pob txha

Prostate kev nyab xeeb: Cuam tshuam kev ua si hauv cov nqaij mos

Zoo heev Anabolic:

Nce cov nqaij ntshiv lub cev loj: Cov kev tshawb fawb soj ntsuam tau pom tias muaj qhov qhib - Nyob rau hauv cov nqaij ntshiv lub cev

Lub Zog Li: Txhim kho cov leeg nqaij thiab lub zog thiab kev ua kis las

Pob Txha Kev Noj Qab Haus Huv: Nce pob txha ceev thiab txhim kho pob txha ua tau zoo

Cov yam ntxwv nyab xeeb:

Hypoandrogenicity: Tsawg Txiaj Fwv ntawm Androgenic phiv

Tsis muaj kev sib cav: Tsis muaj hloov dua siab tshiab rau estrogen, tsis muaj kev pheej hmoo ntawm dej rov qab

Tsawg Hepatotoxicity: Zoo zam los ntawm daim siab ntawm kho cov koob tshuaj


Cov kev siv raws tu qauv

1. Kev Tshawb Fawb Txog Kev Tshawb Fawb:

Pib koob tshuaj:

1 mg ib zaug txhua hnub

Kev Ntsuam Xyuas Kev Ntsuas Rau 1 Lub Limtiam

Escalating koob tshuaj:

Lim tiam 2: 2 mg / hnub

Los ntawm 3 lub lim tiam dhau los: kho rau 3-5 mg / hnub raws li kev kawm xav tau

Koob tshuaj ntau tshaj plaws:

Qhov kev kawm dose tsis tshaj 10 mg / hnub

2. Siv kev voj voog:

Luv - lus kawm: 4-6 lub lis piam

Ntev - lub sij hawm kawm: 8-12 lub lis piam (yuav tsum muaj kev soj ntsuam ze)

Tshaj tawm - kev mus kuaj xyuas: Txuas ntxiv saib xyuas 4 lub lis piam tom qab siv tshuaj noj

3. Saib xyuas cov ntsuas:

Cov hauj lwm ua hauj lwm zoo​:

Hloov pauv ntawm cov nqaij ntshiv lub cev

Cov leeg ua kom muaj zog kuaj

Kev Ntsuas Pob Txom

Qhov ntsuas kev nyab xeeb:

Daim Siab Ua Haujlwm Kev Ntsuam Xyuas

Cov qib ntshav lipid

Hormone Qib Kev Ntsuam Xyuas


Vim li cas thiaj xaiv LGD-4033 cov khoom siv raw?

Siab Xaiv: Muaj kev xaiv thiab muaj kev sib cav heev rau Androgen Receptors

Cov leeg muaj zog: Cov kev tshawb fawb soj ntsuam tau ua pov thawj qhov tseem ceeb nce nyob rau hauv cov nqaij ntshiv lub cev thiab cov leeg kom muaj zog

Kev tshawb nrhiav tus nqi: Nws muaj cov tseem ceeb tshawb fawb hauv kev kho mob ntawm cov leeg leeg atrophy thiab osteoporosis


Lub ntsiab

LGD-4033 yogIb qho cuab yeej tseem ceeb hauv kev tshawb fawb ntawm kev xaiv cov androgen receptor modulators.DhauKev tshawb fawb txuj ci txheej txheem,Nws tuaj yeem tsim rau hauvNtau cov ntaub ntawv muab tshuaj, suav nrog cov ntsiav tshuaj ntawm qhov ncaujCov. Xaiv peb kom ntseeg tausiab -} Purity raw cov ntaub ntawv, kev txhawb nqa kev ua haujlwm, thiab muaj txhij txhua {{1} kev pab muag khoom.


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