Yk {11 10 mg * 100 / Lub raj mis Stromusc Qhov Muag

Yk {11 10 mg * 100 / Lub raj mis Stromusc Qhov Muag
Khoom Taw qhia:
YK11, ib qho tshiab steroid- sarm hypertration thiab qia cell prottration los ntawm inhibiting myostatin thiab ua kom zoo nkauj Androgen receptors. Cov kev tshawb fawb tau pom tias nws muaj peev xwm kov yeej cov leeg nqaij cuam tshuam, thaum tshawb pom cov kev pheej hmoo ntawm estrogen hloov dua siab tshiab.
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Hauj lwm lawm
Kev tsis

Yk11 (Myostatin inhibitor) 10mg 100 ntsiav tshuaj / cov ntaub ntawv hauv lub mis*

Kws Tshuaj Kho Mob - qib ua yeeb|Yk11 (thawj myostatin inhibitor sarm)

Tshuaj lom neeg npe: (2s, 3s, 5s, 10r, 13s, 17s)- 17 - [(1R) -1,2,3-cyclopentane-10,13 -Dimethyl-2,3,4,5,11,12,14,15,16-decahydro-1h-cyclopenta [a] phenanghenhe-17-ol

Tus lej: 431579-34-9

Molecular Cov Qauv: C₃₀h₄₄o₃

Molecular hnyav: 452.68

Cov Lus Qhia Tshwj Xeeb: 10mg / ntsiav tshuaj, 100 ntsiav tshuaj / Lub raj mis

Dosage Daim Ntawv: Enteric - co ntsiav tshuaj

Zog: Dawb Enteric - co ntsiav tshuaj nrog cov kab sib faib


Cov teebmeem tseem ceeb

Yk11 yog aThawj -} hauv-}}} Chav Kawm Xaiv Androgen Receptor Modulator (SRM) ntawm Myostatin Inhibitor ClassCov. Vim nwsTxawv txawv Ob Txhais Txheej Txheem, nws yog dav siv rauCov leeg nqaij loj hlob, lub zog sib zog, thiab kev ua tau huab ua kom zoo nkauj.

Dual kev nqis tes:

Myostatin inhibition: Ncaj qha inhibits myostatin, tshem tawm cov kev txwv ntawm cov leeg loj hlob

Androgen receptor kev cai: Xaiv cov kev ua kom tau txais cov khoom siv Androgenors los txhawb cov protein synthesis

Synergistic cuam tshuam: Dual Txoj kev uas ua tiav cov leeg tau los ntawm cov leeg kev loj hlob dhau ib txwm sarms

Qhov kawg cov leeg nqaij - eints:

Cov leeg tub rog: Xauv lub ntuj kev txwv ntawm myostatin ntawm cov leeg kev loj hlob

MyOfiber hyperplasia: Txhawb kev nce ntxiv nyob rau hauv tus naj npawb ntawm cov leeg nqaij fibers (hyperplasia)

Kev sib zog ua rau muaj zog: Cov Tub Ntxhais Zog Zog Ua Ntej tau nce los ntawm 30-50%

Cov khoom lag luam metabolic tshwj xeeb:

Ensally nquag: Siab bioavailability, tsis muaj kev txhaj tshuaj

Luv ib nrab - lub neej: Txog 2-4 teev, xav tau kev faib khoom noj

Tsis muaj kev sib cav: Tsis muaj hloov dua siab tshiab rau estrogen, tsis muaj kev pheej hmoo ntawm dej rov qab

Qhov Zoo:

Ua txhaum lub physiological txwv: Xauv ntuj txwv rau cov leeg kev loj hlob

Dual kev txiav txim: myostatin inhibition + androgen receptor ua kom tiav

Cov leeg muaj zog: Outperforming cov tsoos sarms


Kawg Cov Khoom Qhia Khoom Siv Khoom Taw Qhia

1. Kev npaj ntawm interic - coated ntsiav tshuaj (10 mg / ntsiav tshuaj):

Piv Txwv Piv Txwv(rau 1000 ntsiav tshuaj):

Yk11 raw khoom: 10.0g

Microcrystalline Cellulose: 80.0g

Lactose: 50.0g

Hla -} Txuas cov carboxymethyl cellulose sidium: 8.0g

Magnesium Stearate: 2.0g

Npaj txheej txheem:

Cov Khoom Siv Raw Ua Ntej: Micronization (D90 tsawg dua los yog sib npaug rau 10μm)

Cov nqi sib xyaw sib xyaw: maj mam sib tov nrog rau dituent

Ntub av granulle: Granulate nrog cov nyiaj uas tsim nyog ntawm cov dej huv thiab qhuav hauv cov kua hauv 50 degree

Granulation: 20 Mesh Sab Canules, ntxiv Flow AIDS thiab roj nplua nyeem

Ntsiav tshuaj: 8mm round tuag, 8-10kn siab ntsiav tshuaj

Enteric Txheej:) PH {{- Nyob Ntawm Txoj Kev Nkag Mus Rau Txoj hnyuv Tso Tawm

Kev Tswj Xyuas Zoo:

Cov ntsiab lus sib xyaw: RSD tsawg dua lossis sib npaug rau 3% (HPLC Nrhiav tau)

Kev tshem tawm: Tsawg dua lossis sib npaug nrog 10% hauv cov kua txiv pais plab tsis pub dhau 2 teev, ntau dua lossis sib npaug hauv cov kua txob hauv plab tsis pub dhau 45 feeb

Lwm yam tshuaj: Ib leeg impurity tsawg dua los yog sib npaug rau 0.5%, tag nrho cov impurities tsawg dua los yog sib npaug rau 1.0%

2. Npaj sau ntawv:

Noo noo - pov thawj kev kho mob: Cov khoom siv raw yog hygroscopic thiab amrient vos yuav tsum tau tswj hwm

Lub teeb -} Cov ntaub ntawv ua haujlwm: nkag siab lub teeb, yuav tsum tau ntim rau hauv ib lub teeb -}} eutshu

Enteric coated lav: Kom tsis txhob muaj kev sib cais hauv lub plab thiab tsom rau hauv txoj hnyuv


Cov kev siv raws tu qauv

1. Txheem kev siv cov xwm txheej:

Ntse Didimen:

Pib koob tshuaj: 5 mg ob zaug ib hnub

Txij Nkawm Dose: 10 mg ob zaug ib hnub

Qhov tshuaj ntau tshaj plaws: tsis muaj ntau tshaj 30 mg / hnub

Voj voog ntev​:

Txheem Ciaje: 4-6 lub lis piam

Advanced Cycle: 6-8 lub lis piam (yuav tsum tau soj ntsuam ze)

2. Sib cais - dose dosing lub tswv yim:

Dose lub sij hawm:

Sawv ntxov: Siv sijhawm 1 teev ua ntej kev qhia ua ntej

Yav tsaus ntuj: Noj tom qab kev cob qhia lossis ua ntej txaj

Noj ntawm lub plab khoob: Noj 1 teev ua ntej lossis 2 teev tom qab noj mov

3. Kev siv nyiaj siab:

Kev Cuam Tshuam​:

Dosage: 10 mg peb zaug ib hnub

Lub Sij Hawm: 4 lub lis piam (nce siab heev)

Tu voj voog txij nkawm:

Dosage: 5 mg ob zaug ib hnub

Lub Sij Hawm: 4-6 lub lis piam (sib sau ua ke)

4. Post -} kev voj voog kev kho (PCT):

Pct tsis muaj:

Txhua tus yk11 cycles yuav tsum tau ua raws PCT

Muaj zog inhibit endogenous Testosterone zais cia

CCT program:

Tamoxifen: 20 mg / hnub rau 4 lub lis piam

Clomiphene: 50 mg / hnub rau 2 lub lis piam, 25 mg / hnub rau 2 lub lis piam

5. Txheej Txheem Tswjhwm:

Cov kev mob tshwm sim ntau:

Nruj nreem hauv cov pob qij txha (vim cov leeg mob sai)

Nce cov leeg siab

Muaj zog inhibition ntawm HTTA axis

Countermeasures:

Pab Txhawb Ntxiv Cov Tiv Thaiv (Glucosamine, Chondroitin)

Kev Kawm Kom Zoo Dua

Nruj me ntsis nqa pcct


Vim li cas thiaj xaiv Yk11?

Myostatin inhibition: Tsuas yog SEARM uas ncaj qha tiv thaiv cov leeg txoj kev loj hlob cuam tshuam

Dual kev nqis tes: Ua txhaum los ntawm kev txwv ntawm cov leeg nqaij -}} Siv tshuaj

Cov leeg muaj zog loj hlob: Ua tiav cov leeg kev loj hlob dhau lub cev txwv


Kev Muaj Peev Xwm Zoo:

CGMP Txuj Ci Ntau Lawm: Kev tswj hwm nruj zoo

Cov ntaub ntawv muaj kev ruaj khov: Kuaj tau nrawm rau 6 lub hlis sib ntsib cov qauv

Thib peb -} Kev Ntsuas Cov Lus Qhia: Coa daim ntawv pov thawj yog muab rau txhua pob

Kev Ntim:

Noo noo -} ntawv pov thawj fwj: 100 ntsiav tshuaj / lub raj mis, ua - hauv desiccant

Lub teeb -} ntaub ntawv tiv thaiv: Aluminium-} Yas blister + Lub Teeb - eCEFEF POLTEJ OB CHAV tiv thaiv

Cap: Tiv thaiv cov menyuam yaus los ntawm kev nqos tsis tau


Tag

Yk11 yogA nroos moov hipsatin inhibitor sharm cov khoom, tshwj xeeb haum rauCov neeg siv khoom tau nrhiav cov leeg nqaij loj hlob thiab lub zog sib zogCov. Cov koob tshuaj pom zoo yog10-20mg / hnub rau 4-6Lub voj voog lub voj voog.

Xav tau txoj kev npaj tus kheej lub voj voog?

Peb muab cov tshuaj qhia kev tshaj lij los pab koj siv cov khoom kom nyab xeeb thiab ua kom zoo!


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Cim npe nrov: yk {11 10 mg * 100 / lub raj mis Stromusc qhov ncauj, Tuam Tshoj

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