Selank 5mg / lub raj mis kev taw qhia
Pharmaceutical -qib peptide formulations|Ua nyob rau hauv Suav teb los ntawm Selank
Tshuaj npe: Thr-Lys-Pro-Arg-Pro-Gly-Pro
Ib ntus: TKPRGP
CAS Nr.: 129954-34-3
Specification: 5mg / lub raj mis
Daim ntawv noj tshuaj: Lyophilized hmoov rau kev txhaj tshuaj
Cov mis mos molecular: C₃₃H₅₇N₁₁O₉
Molecular hnyav: 751.89
Qhov tshwm sim: Dawb khov- cov hmoov qhuav qhuav
Purity: Ntau dua lossis sib npaug li 98% (HPLC kuaj pom)
Cia tej yam kev mob: Khaws ntawm -20℃deb ntawm lub teeb.
Cov teebmeem tseem ceeb
Seranc yog ibhluavtaws heptapeptidenrogtiv thaiv -kev ntxhov siab, neuroprotective thiab kev txawj ntse- txhim kho cov teebmeem, thiab yog dav siv nyob rau hauvkev kho mob ntawm kev ntxhov siab, kev txhim kho kev nco thiab kev tshawb fawb txog cov kab mob neurodegenerative.
✅ Ntau yammechanisms ntawm kev ua:
GABA txoj cai: Influences GABAergic system, txo kev ntxhov siab.
Nce qib BDNF: Txhim kho lub hlwb- tau txais txiaj ntsig neurotrophic (BDNF) qib.
Kev tiv thaiv kab mob: tswj cytokines thiab ntsuas lub cev tiv thaiv kab mob.
✅Qualityqhov zoo ntawm Suav manufacturing:
Purity Guaranteed: Khoom-theem synthesis txheej txheem, purity Ntau dua los yog sib npaug rau 98%, ib qho impurities Tsawg dua los yog sib npaug rau 0.1%.
Ua raws li qhov tseeb: Heptapeptide ib ntus 100% raug
Kev pom zoo ua haujlwm: In vitro BDNF assay EC50=0.1 nM
✅ thoob ntiaj tebmuab kev ruaj ntseg:
Cold chain logistics: -20℃txias saw tsheb thauj mus los thoob plaws tag nrho cov txheej txheem los xyuas kom meej cov khoom ruaj khov.
Ntau- khoom xa tuaj: Cov tsev khaws khoom hauv cheeb tsam tau tsim nyob rau hauv Suav teb, Tebchaws Europe, Amelikas, thiab Asia - cheeb tsam Pacific, ua kom cov khoom xa tuaj hauv 7 hnub.
Kev them nyiaj yug kev lis kev cai clearance: Kev npaj cov ntaub ntawv ua kom muaj kev lis kev cai zoo thoob ntiaj teb.
Cov txheej txheem ntau lawm thiab kev ruaj ntseg zoo
1. Advanced synthesis txheej txheem:
Khoom -phase synthesis: The Fmoc solid-phase synthesis strategy was adopted, with a condensation efficiency >99.5%.
Kev ua kom huv huv: Npaj HPLC purification, gradient elution, sau ntawm lub ntsiab ncov.
Txias- tshuab ziab khaub ncaws: kub- tswj khov- ziab, cov ntsiab lus noo noo tsawg dua lossis sib npaug li 3.0%.
2. Cov qauv kev tswj xyuas nruj:
Tshuaj purity:
Cov ntsiab lus tseem ceeb: 98.0% ~ 102.0%
Cov khoom muaj feem xyuam: Ib qho impurity Tsawg dua lossis sib npaug li 0.1%, tag nrho impurities Tsawg dua lossis sib npaug li 0.5%
Cov ntsiab lus acetic acid: tsawg dua lossis sib npaug li 10.0% (ion chromatography)
Kev ua si lom neeg:
Kev sim ntawm tes: BDNF qhia tau nce los ntawm tsawg kawg 90% piv rau tus qauv.
Kev sim tsiaj: Tiv thaiv-kev ntxhov siab ED50=0.3 mg/kg
3. Cov ntaub ntawv ruaj ntseg:
Ntev -lub sij hawm ruaj khov: Khaws ntawm -20℃rau 24 lub hlis, txhua qhov ntsuas tau ua tau raws li qhov xav tau.
Kev ntsuas nrawm: Tom qab khaws cia ntawm 25℃rau 6 lub hlis, purity txo qis dua los yog sib npaug li 2.0%.
Kev ruaj ntseg hauv kev siv: Tom qab rov kho dua, khaws cia ntawm 2-8℃rau 7 hnub; purity Ntau dua lossis sib npaug li 95%.
Kev Tshawb Fawb Txog Kev Tshawb Fawb thiab Kev Tshawb Fawb Txog Kev Tshawb Fawb
1. Mechanism ntawm kev kawm ua:
Neuroprotection: Tiv thaiv neurons los ntawm txoj kev BDNF
Kev ntxhov siab: Kev tswj hwm GABA kom txo cov kev ntxhov siab
Txhim khu kev nco: Txhim kho kev kawm thiab kev nco muaj peev xwm
2. Kev tshawb fawb thiab kev siv thaj chaw:
Kev puas hlwb: Kev Tshawb Fawb Txog Kev Kho Mob Generalized Anxiety Disorder thiab Post-Taumatic Stress Disorder
Neuroscience: Kev Tshawb Fawb Neuroprotective hauv Alzheimer's thiab Parkinson's Diseases
Kev txawj ntse: Kev Tshawb Fawb Txog Kev Kawm thiab Me Me Mechanisms thiab Txhim Kho
3. Preclinical cov ntaub ntawv:
Kev ntxhov siab txog kev txhim kho: Tsiaj cov kev tshawb fawb qhia tau hais tias 40-60% txo tus cwj pwm ntxhov siab.
Txhim Kho Kev Nco: Txhim kho qhov tseem ceeb hauv Spatial thiab ua haujlwm nco
Zoo kev nyab xeeb profile: dav kho qhov rais, tsis tshua muaj kev pheej hmoo ntawm kev phiv.
Tuam Tshoj txoj kev tsim khoom zoo
1. Qhov zoo ntawm kev tsim khoom:
Synthesis technology: Microwave-pab khoom- lub xeev synthesis nrog kev ua kom muaj kuab paug siab.
Kev ua kom huv huv: Preparative HPLC purification, purity Ntau dua lossis sib npaug li 98%.
Kev tswj kom zoo: Kev tswj xyuas zoo thoob plaws tag nrho cov txheej txheem los ntawm cov khoom siv raw mus rau cov khoom tiav.
2. Kev Tswj Xyuas Zoo:
Ua raws li cov qauv: Ua tau raws li Suav Pharmacopoeia, USP, thiab EP cov qauv.
Kev kawm ruaj khov: Ua kom tiav kev tshawb nrhiav kev ruaj ntseg.
Batch sib xws: Cov txheej txheem nruj tswj xyuas kom zoo sib xws ntawm cov khoom siv.
3. Ntiaj teb no mov network:
Lub hauv paus tsim: GMP-raws li kev tsim khoom hauv Suav teb
Kev faib tawm network: Lub thoob ntiaj teb kev faib khoom thiab cov saw hlau txias logistics network
Kev them nyiaj yug rau npe: Txhawb cov ntawv sau npe los ntawm cov teb chaws thoob ntiaj teb.
Vim li cas thiaj xaiv Suav - ua Seranke ?
Ntaucov txiaj ntsig: Los tiv thaiv-kev ntxhov siab, kev tiv thaiv neuroprotective, thiab kev paub txog kev txawj ntse
Siabkev huv: Tshaj 98% purity, nrog kev tswj xyuas nruj.
Activekev paub tseeb: Kev sim tsiaj txhu pom ED50 ntawm 0.3 mg / kg, qhia tias muaj zog.
ruaj khovmuab: Ib qho kev xa khoom tiav ua kom muaj kev xa khoom raws sij hawm thiab txhim khu kev qha.
Cov ntsiab lus
Ua nyob rau hauv Suav teb, Seranc 5mg lyophilized hmoov rau txhajsawv cev rau siab - tus qauv zoo ntawm neuromodulatory peptides. Los ntawmcov txheej txheem synthesis siab heev, kev tswj xyuas kom zoo, thiab cov khoom siv ruaj khov, nws muabsiab -zoo, cov cuab yeej tshawb fawb zoo heev rau kev tshawb fawb thoob ntiaj teb ntawm cov kab mob neuropsychiatric. Xaiv Ua hauv Suav teb txhais tau tias xaivkev tshawb fawb-qib zoo thiab txhim khu kev qha.
Need dab tsi, thov hu raupeb
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