Epitalon 10mg / lub raj mis qhia
Pharmaceutical -qib peptide formulations|Ua nyob rau hauv Suav teb, Epitalon
Tshuaj npe: L-alanyl-L-glutamyl-L-asparaginyl-L-glycine
Ib ntus: Ala-Glu-Asp-Gly
CAS Nr.: 307297-39-8
Specification: 10mg / lub raj mis
Daim ntawv noj tshuaj: Lyophilized hmoov rau kev txhaj tshuaj
Cov mis mos molecular: C₁₄H₂₂N₄O₈
Molecular hnyav: 390.35
Qhov tshwm sim: Dawb khov- cov hmoov qhuav qhuav
Purity: Ntau dua lossis sib npaug li 98% (HPLC kuaj pom)
Cia tej yam kev mob: Khaws ntawm -20℃deb ntawm lub teeb.
Cov teebmeem tseem ceeb
Aptamethasone yog atelomerase - qhib tetrapeptideuas yog dav siv nyob rau hauvanti- tshawb fawb kev laus, telomere biology, thiab hnub nyoog-kev tshawb fawb txog kab mobvim nwstshwj xeeb telomere tu thiab tiv thaiv -aging zog.
✅Tsimkho mechanism:
Telomerase activation: Upregulates telomerase kev ua ub no thiab prolongs telomere ntev.
Cellular senescence: Ncua cell replication thiab senescence, extending cell lifespan
Gene stability: Tswj chromosome stability thiab txo DNA puas
✅Qualityqhov zoo ntawm Suav manufacturing:
Purity Guaranteed: Khoom-theem synthesis txheej txheem, purity Ntau dua los yog sib npaug rau 98%, ib qho impurities Tsawg dua los yog sib npaug rau 0.1%.
Ua raws li qhov tseeb: Tetrapeptide ib ntus 100% raug
Kev pom zoo ua haujlwm: Cellular telomerase kev ua haujlwm nce 3-5 zaug.
✅ thoob ntiaj tebmuab kev ruaj ntseg:
Cold chain logistics: -20℃txias saw tsheb thauj mus los thoob plaws tag nrho cov txheej txheem los xyuas kom meej cov khoom ruaj khov.
Ntau- khoom xa tuaj: Cov tsev khaws khoom hauv cheeb tsam tau tsim nyob rau hauv Suav teb, Tebchaws Europe, Amelikas, thiab Asia - cheeb tsam Pacific, ua kom cov khoom xa tuaj hauv 7 hnub.
Kev them nyiaj yug kev lis kev cai clearance: Kev npaj cov ntaub ntawv ua kom muaj kev lis kev cai zoo thoob ntiaj teb.
Cov txheej txheem ntau lawm thiab kev ruaj ntseg zoo
1. Advanced synthesis txheej txheem:
Khoom -phase synthesis: The Fmoc solid-phase synthesis strategy was adopted, with a condensation efficiency >99.5%.
Kev ua kom huv huv: Npaj HPLC purification, gradient elution, sau ntawm lub ntsiab ncov.
Txias- tshuab ziab khaub ncaws: kub- tswj khov- ziab, cov ntsiab lus noo noo tsawg dua lossis sib npaug li 3.0%.
2. Cov qauv kev tswj xyuas nruj:
Tshuaj purity:
Cov ntsiab lus tseem ceeb: 98.0% ~ 102.0%
Cov khoom muaj feem xyuam: Ib qho impurity Tsawg dua lossis sib npaug li 0.1%, tag nrho impurities Tsawg dua lossis sib npaug li 0.5%
Cov ntsiab lus acetic acid: tsawg dua lossis sib npaug li 10.0% (ion chromatography)
Kev ua si lom neeg:
Kev sim ntawm tes: Telomerase kev ua haujlwm tau nce tsawg kawg 90% piv rau tus qauv.
Tsiaj sim: Lifespan txuas ntxiv los ntawm 15-20%
3. Cov ntaub ntawv ruaj ntseg:
Ntev -lub sij hawm ruaj khov: Khaws ntawm -20℃rau 24 lub hlis, txhua qhov ntsuas tau ua tau raws li qhov xav tau.
Kev ntsuas nrawm: Tom qab khaws cia ntawm 25℃rau 6 lub hlis, purity txo qis dua los yog sib npaug li 2.0%.
Kev ruaj ntseg hauv kev siv: Tom qab rov kho dua, khaws cia ntawm 2-8℃rau 7 hnub; purity Ntau dua lossis sib npaug li 95%.
Kev Tshawb Fawb Txog Kev Tshawb Fawb thiab Kev Tshawb Fawb Txog Kev Tshawb Fawb
1. Mechanism ntawm kev kawm ua:
Telomere kev saib xyuas: Telomere ntev yog tswj los ntawm kev ua kom telomerase.
Anti- laus: Txo cov txheej txheem cellular aging thiab ncua kev noj qab haus huv lifespan.
Gene stability: Ua kom ruaj khov genome thiab txo qis kev hloov pauv.
2. Kev tshawb fawb thiab kev siv thaj chaw:
Kev Tshawb Fawb Txog Kev Laus: Kawm txog Cellular Senescence Mechanisms thiab Intervention Strategies
Oncology: Kev Tshawb Fawb Txog Kev Sib Raug Zoo ntawm Telomere Length thiab Tumor Development
Cov kab mob degenerative: Kev tshawb fawb txog kev tiv thaiv thiab kev kho mob hnub nyoog -txog kab mob
3. Preclinical cov ntaub ntawv:
Extended lifespan: Tsiaj thwmsim qhia qhov nruab nrab lifespan nce ntawm 15-20%.
Kev txhim kho kev noj qab haus huv: Txo qhov tshwm sim ntawm lub hnub nyoog -txog kab mob
Zoo kev nyab xeeb profile: dav kho qhov rais, tsis tshua muaj kev pheej hmoo ntawm kev phiv.
Tuam Tshoj txoj kev tsim khoom zoo
1. Qhov zoo ntawm kev tsim khoom:
Synthesis technology: Microwave-pab khoom- lub xeev synthesis nrog kev ua kom muaj kuab paug siab.
Kev ua kom huv huv: Preparative HPLC purification, purity Ntau dua lossis sib npaug li 98%.
Kev tswj kom zoo: Kev tswj xyuas zoo thoob plaws tag nrho cov txheej txheem los ntawm cov khoom siv raw mus rau cov khoom tiav.
2. Kev Tswj Xyuas Zoo:
Ua raws li cov qauv: Ua tau raws li Suav Pharmacopoeia, USP, thiab EP cov qauv.
Kev kawm ruaj khov: Ua kom tiav kev tshawb nrhiav kev ruaj ntseg.
Batch sib xws: Cov txheej txheem nruj tswj xyuas kom zoo sib xws ntawm cov khoom siv.
3. Ntiaj teb no mov network:
Lub hauv paus tsim: GMP-raws li kev tsim khoom hauv Suav teb
Kev faib tawm network: Lub thoob ntiaj teb kev faib khoom thiab cov saw hlau txias logistics network
Kev them nyiaj yug rau npe: Txhawb cov ntawv sau npe los ntawm cov teb chaws thoob ntiaj teb.
Vim li cas thiaj xaiv Aipatai, cov khoom lag luam hauv Suav teb?
Anti-kev laus pioneer: Thawj hluavtaws peptide pov thawj kom ntev telomere
Siabkev huv: Tshaj 98% purity, nrog kev tswj xyuas nruj.
Ua komkev lees paub: Telomerase kev ua haujlwm hauv hlwb nce 3-5 zaug
ruaj khovmuab: Ib qho kev xa khoom tiav ua kom muaj kev xa khoom raws sij hawm thiab txhim khu kev qha.
Cov ntsiab lus
Ua nyob rau hauv Suav teb, Aipatet 10mg lyophilized hmoov rau txhajsawv cev rau qib siab - qauv zoo rau telomere biology tshawb fawb cov cuab yeej. Los ntawmadvanced synthesis txheej txheem, nruj zoo tswj, thiab ib tug ruaj khov mov system,nws muabsiab -cov cuab yeej tshawb fawb zoo heevrauthoob ntiaj teb kev tiv thaiv- laus thiab hnub nyoog- kev tshawb fawb txog kab mob. Xaiv Ua hauv Suav teb txhais tau tias xaivkev tshawb fawb-qib zoo thiab txhim khu kev qha.
Need dab tsi, thov hu raupeb
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