DSIP 2mg / lub raj mis qhia
Pharmaceutical -qib peptide formulation|Delta Pw tsaug zog-Inducing Peptide, ua nyob rau hauv Suav teb
Tshuaj npe: Tryptophanyl-alanyl-glycyl-glycyl-aspartyl-alanyl-seryl-glycyl-glutamic acid
Ib ntus: H-Trp-Ala-Gly-Gly-Asp-Ala-Ser-Gly-Glu-OH
CAS Nr.: 62568-57-4
Specification: 2mg / lub raj mis
Daim ntawv noj tshuaj: Lyophilized hmoov rau kev txhaj tshuaj
Cov mis mos molecular: C₃₄H₄₇N₁₁O₁₇
Molecular hnyav: 849.80
Qhov tshwm sim: Dawb khov- cov hmoov qhuav qhuav
Purity: Ntau dua lossis sib npaug li 98% (HPLC kuaj pom)
Cia tej yam kev mob: Khaws ntawm -20℃deb ntawm lub teeb.
Cov teebmeem tseem ceeb
DSIP yog ib qhoendogenous neuropeptideuas yog dav siv nyob rau hauvkev kho mob ntawm kev pw tsaug zog, kev tshawb fawb neuroprotective, thiab circadian atherosclerosis tswjvim nwstshwj xeeb kev cai pw tsaug zog muaj nuj nqi thiab neuroprotective zog.
✅ pw tsaug zogkev cai mechanism:
Pw tsaug zog induction: Txhawb qeeb-yoj pw tsaug zog thiab ua kom lub sijhawm pw tsaug zog.
Neuroprotection: Txo cov tshuaj hormones kev ntxhov siab thiab tiv thaiv cov neurons los ntawm kev puas tsuaj.
Circadian atherosclerosis kev cai: Tswj lub moos lom neeg thiab txhim kho kev pw tsaug zog -Wake cycle.
✅Qualityqhov zoo ntawm Suav manufacturing:
Purity Guaranteed: Khoom-theem synthesis txheej txheem, purity Ntau dua los yog sib npaug rau 98%, ib qho impurities Tsawg dua los yog sib npaug rau 0.1%.
Ua raws li qhov tseeb: Cov kab mob nonapeptide yog 100% raug.
Kev lees paub ntawm kev ua haujlwm: ED50=0.1 mg/kg hauv kev sim pw tsaug zog tsiaj.
✅ thoob ntiaj tebmuab kev ruaj ntseg:
Cold chain logistics: -20℃txias saw tsheb thauj mus los thoob plaws tag nrho cov txheej txheem los xyuas kom meej cov khoom ruaj khov.
Ntau- khoom xa tuaj: Cov tsev khaws khoom hauv cheeb tsam tau tsim nyob rau hauv Suav teb, Tebchaws Europe, Amelikas, thiab Asia - cheeb tsam Pacific, ua kom cov khoom xa tuaj hauv 7 hnub.
Kev them nyiaj yug kev lis kev cai clearance: Kev npaj cov ntaub ntawv ua kom muaj kev lis kev cai zoo thoob ntiaj teb.
Cov txheej txheem ntau lawm thiab kev ruaj ntseg zoo
1. Advanced synthesis txheej txheem:
Khoom -phase synthesis: The Fmoc solid-phase synthesis strategy was adopted, with a condensation efficiency >99.5%.
Kev ua kom huv huv: Npaj HPLC purification, gradient elution, sau ntawm lub ntsiab ncov.
Txias- tshuab ziab khaub ncaws: kub- tswj khov- ziab, cov ntsiab lus noo noo tsawg dua lossis sib npaug li 3.0%.
2. Cov qauv kev tswj xyuas nruj:
Tshuaj purity:
Cov ntsiab lus tseem ceeb: 98.0% ~ 102.0%
Cov khoom muaj feem xyuam: Ib qho impurity Tsawg dua lossis sib npaug li 0.1%, tag nrho impurities Tsawg dua lossis sib npaug li 0.5%
Cov ntsiab lus acetic acid: tsawg dua lossis sib npaug li 10.0% (ion chromatography)
Kev ua si lom neeg:
Pw tsaug zog induction test: potency tsis tsawg dua 90% ntawm tus qauv.
Electroencephalogram (EEG) test: Ua tau raws li cov qauv zoo
3. Cov ntaub ntawv ruaj ntseg:
Ntev -lub sij hawm ruaj khov: Khaws ntawm -20℃rau 24 lub hlis, txhua qhov ntsuas tau ua tau raws li qhov xav tau.
Kev ntsuas nrawm: Tom qab khaws cia ntawm 25℃rau 6 lub hlis, purity txo qis dua los yog sib npaug li 2.0%.
Kev ruaj ntseg hauv kev siv: Tom qab rov kho dua, khaws cia ntawm 2-8℃rau 7 hnub; purity Ntau dua lossis sib npaug li 95%.
Kev Tshawb Fawb Txog Kev Tshawb Fawb thiab Kev Tshawb Fawb Txog Kev Tshawb Fawb
1. Mechanism ntawm kev kawm ua:
Kev cai pw tsaug zog: tshwj xeeb txhawb nqa delta-yoj lub hlwb ua haujlwm
Neuroprotection: Txo cov qib cortisol thiab txo kev ntxhov siab.
Lub suab synchronization: Tswj cov kev ua ntawm suprachiasmatic nucleus thiab synchronizes lom rhythms.
2. Kev tshawb fawb thiab kev siv thaj chaw:
Pw Tshuaj: Kev Tshawb Fawb Txog Kev Kho Mob Insomnia thiab Pw Tsaug Zog Tsis Txaus Siab
Neuroscience: Kev Tshawb Fawb Txog Kev Tiv Thaiv Kev Tiv Thaiv Cov Kab Mob Neurodegenerative
Kev puas hlwb: Kev tshawb fawb txog kev kho mob ntxiv rau kev ntxhov siab thiab kev nyuaj siab
3. Preclinical cov ntaub ntawv:
Kev pw tsaug zog zoo dua: Tsiaj cov kev tshawb fawb pom tias 50-70% nce hauv kev pw tsaug zog qeeb.
Kev tiv thaiv kev ntxhov siab: Qhov tseem ceeb txo qis cov tshuaj hormones
Zoo kev nyab xeeb profile: dav kho qhov rais, tsis tshua muaj kev pheej hmoo ntawm kev phiv.
Tuam Tshoj txoj kev tsim khoom zoo
1. Qhov zoo ntawm kev tsim khoom:
Synthesis technology: Microwave-pab khoom- lub xeev synthesis nrog kev ua kom muaj kuab paug siab.
Kev ua kom huv huv: Preparative HPLC purification, purity Ntau dua lossis sib npaug li 98%.
Kev tswj kom zoo: Kev tswj xyuas zoo thoob plaws tag nrho cov txheej txheem los ntawm cov khoom siv raw mus rau cov khoom tiav.
2. Kev Tswj Xyuas Zoo:
Ua raws li cov qauv: Ua tau raws li Suav Pharmacopoeia, USP, thiab EP cov qauv.
Kev kawm ruaj khov: Ua kom tiav kev tshawb nrhiav kev ruaj ntseg.
Batch sib xws: Cov txheej txheem nruj tswj xyuas kom zoo sib xws ntawm cov khoom siv.
3. Ntiaj teb no mov network:
Lub hauv paus tsim: GMP-raws li kev tsim khoom hauv Suav teb
Kev faib tawm network: Lub thoob ntiaj teb kev faib khoom thiab cov saw hlau txias logistics network
Kev them nyiaj yug rau npe: Txhawb cov ntawv sau npe los ntawm cov teb chaws thoob ntiaj teb.
Vim li cas thiaj xaiv DSIP tsim nyob rau hauv Suav teb?
Endogenoustshuaj: Pw tsaug zog- tswj peptides ib txwm muaj nyob hauv tib neeg lub cev
Siabkev huv: Tshaj 98% purity, nrog kev tswj xyuas nruj.
Activekev paub tseeb: Tsiaj thwmsim pom ED50 ntawm 0.1 mg/kg, qhia tau hais tias muaj zog.
ruaj khovmuab: Ib qho kev xa khoom tiav ua kom muaj kev xa khoom raws sij hawm thiab txhim khu kev qha.
Cov ntsiab lus
Ua nyob rau hauv Suav teb, DSIP 2mg lyophilized hmoov rau txhajsawv cev rau qib siab - qauv zoo ntawm endogenous pw tsaug zog- tswj peptides. Los ntawmcov txheej txheem synthesis siab heev, kev tswj xyuas kom zoo, thiab cov khoom siv ruaj khov, nws muabsiab -zoo, cov cuab yeej tshawb fawb zoo heev rau kev pw tsaug zog thiab kev tshawb fawb txog kev puas siab puas ntsws thoob ntiaj teb. Xaiv Ua hauv Suav teb txhais tau tias xaivkev tshawb fawb-qib zoo thiab txhim khu kev qha.
Xav taudab tsi, thov hu raupeb
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