Hepius hom gw 501516 10 mg 100 cov ntsiav tshuaj tseem ceeb*
Kws Tshuaj Kho Mob - qib ua yeeb|Hepius hom GW501516 (PARP - Δ agonist)
Tshuaj lom neeg npe: 2- (2- (((4-chlorophenyl) (difluoro) methyl) phenoxy) acetamido) acetamide
Cas tsis muaj.: 317318-70-0
Cov Lus Qhia Tshwj Xeeb: 10mg / ntsiav tshuaj, 100 ntsiav tshuaj / Lub raj mis
DOSAGE Daim Ntawv: Zaj duab xis - co ntsiav tshuaj
Molecular cov mis: c₂₁h₁₈f₂n₂o₃s
Molecular hnyav: 416.44
Melting Taw tes: 134-136 Qib
Zog: dawb, cov ntsiav tshuaj hloov nrog sib faib cov kab.
Solubility: me ntsis soluble hauv dej, yooj yim soluble hauv dmo
Purity: ntau dua los yog sib npaug rau 99% (HPLC Nrhiav tau)
Cov teebmeem tseem ceeb
Hepius hom GW501516 yog aKev xaiv siab Proxisome Proliferator -} ™ activ່ວນ receptor delta (ppp- Δ) agonist, dav siv rauKev kho mob ntawm cov metabolic syndrome, kev txhim kho ntawm kev ua kis las, thiab kev txhim kho ntawm kev tswj hwm lub cev vim nws cov kev ua kom zoo nkauj thiab kev ua kom tiav- kev txhim kho kev cuam tshuam.
✅ PPPL - Δ txoj kev ua kom cov yam ntxwv:
Rog oxidation: Ua kom cov kev qhia ntawm fatty acid oxidation genes hauv pob txha pob txha, txhawb nqa cov rog rog.
10 kev kwv yees: Nce cov kev faib ua feem ntawm qeeb - twitch cov leeg nqaij thiab mitochondrial biosynthesis.
Ntshav Ntshav Hmo: Txhim kho cov insulin rhiab heev thiab qab zib audostasis
✅ Hepius Gener Txawv Txawv:
Crystal Daim Ntawv Txhim Kho: Siv ruaj khov -} crystalline raw cov ntaub ntawv, bioavailability yog nce rau 92%.
Yam tshuaj kho: Siv thev naus laus zis Micronization ua kom muaj kev sib luag ntawm cov ntsiab lus nrog RSD tsawg dua lossis sib npaug ntawm 1.0%.
Kev tshwm sim sai sai ntawm kev nqis tes ua: Kev Plasma Peaka Pequma tau mus txog hauv 1 -} 2 teev; Ib nrab-lub neej yog 16-20 teev.
✅ Cov nyhuv metabolic siv tau:
Kev ua kom ntev: Cov kev tshawb fawb preclinical qhia tau 40-50% txhim kho hauv kev ua si kawg kawg.
Rog txo: Tseem ceeb txo lub cev rog feem pua, tshwj xeeb tshaj yog cov rog rog.
Txhim kho cov ntshav lipids: Nce siab - cov lipoprotein me me (HDL) thiab txo qis lipoprotein (LDL).
Hepiev Hom Khoom Zoo Zoo
1. Cov Khoom Siv Raw Khoom Zoo:
Tshuaj lom neeg purity: Raw cov khoom siv ntau dua los yog sib npaug rau 99.5% (HPLC nrhiav tau, zoo dua rau USP qauv)
ISOMER tswj: Txhim kho qhov tseeb configuration ntawm chairal chaw
Cov Kws Koom Tes Tswj: Ib leeg tsis paub tab<0.05%, total impurities <0.1%.
2. Patented tsim tshuab:
Nanoparticle ua: Raw cov ntaub ntawv cov khoom siv me me D90 tsawg dua lossis sib npaug rau 3μm, ua kom muaj kev sib luag sai.
Zov - txheej txheej txheej txheem:
Kev rho tawm txheej: noo noo {{}} Cov ntaub ntawv pov thawj thiab oxidation - ntawv pov thawj
Txhawb nqa - tso txheej txheem: tswj cov nqi tso tawm
Txheej Txheem Tiv Thaiv: Pais plab txheej
Anti -} cov tshuab cuav: Holographic anti -} Counterfeiting daim ntawv, scan code rau txheeb xyuas qhov tseeb.
3. Kev Tsim Kho Ntau Lawm:
Cov ntawv pov thawj thoob ntiaj teb: Tuam Tshoj NMPA GMP ntawv pov thawj, EU GMP qauv
Kev tswj hwm ib puag ncig: Chav ua haujlwm 10,000 kev ntxuav tes, kev saib xyuas ib puag ncig online.
End - rau -}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}} kawg traceazeobility: Ib lub zog hluav taws xob tag nrho cov txheej txheem hluav taws xob tag nrho los ntawm cov khoom raw ua tiav cov khoom tiav.
4. Tswjhwm Saib Xyuas Zoo:
Cov ntsiab lus sib xyaw: RSD tsawg dua lossis sib npaug rau 1.0% (Suav cov tshuaj yuav tsum tau tsawg dua lossis sib npaug rau 6%)
Tus lej sib cais: Loj dua los yog sib npaug rau 90% kev sib nrauj tom qab 30 feeb, ntau dua lossis sib npaug ntawm 95% kev sib nrauj tom qab 45 feeb.
Lwm yam tshuaj: Cov Khoom Ua Phem<0.1%, total impurities <0.2%
Stability: Dhau kev sim ua kom nrawm tom qab 6 lub hlis; Txee lub neej 36 lub hlis.
Hepieve hom preclinical zoo
1. Kev txheeb xyuas qhov tseeb:
Kev txhim kho kom muaj kev txhim kho kev txhim kho: Cov kev tshawb fawb tsiaj qhia pom tias cov kev tawm dag zog thev naus laus zis tuaj yeem nce ntxiv 40-50%.
Kev txhim kho metabolic: Txom Nyem Insulin rhiab heev thiab zoo li kev thev taus
Lub cev muaj pes tsawg leeg: Txo cov roj zuj zus thiab ua kom cov rog rog rog
2. Mechanism ntawm Kev Ua:
Ppp - δ δation: Kev ua kom muaj zog ntawm lub ppp. {}} Δ signing txoj kev
Mitochondrial biosynthesis: Txhawb Mitochondrial tsim thiab fatty acid oxidation.
Ntsuas cov neeg ua pauj: Upregulation ntawm fatty acid oxidation {{}}} Cov noob pom ntsig txog haiv neeg
3. Kev Tshawb Fawb Kev Tshawb Fawb Tus Nqi:
Kev Tshawb Fawb Kab Mob Kev Tshawb Fawb: Kev tshawb fawb ntawm cov txheej txheem ntawm cov kab mob metabolic xws li rog thiab mob ntshav qab zib
Cov Tshuaj Ntaus Tshuaj: Kev tshawb fawb txog kev ua kom muaj kev txhim kho kev ua kom thev taus thiab lub zog metabolism kev cai
Nqaij Metabolism: Kev kawm ntawm pob txha pob txha pob txha litabolism thiab cov kev hloov pauv
Hepius hom kev pabcuam tshaj lij
1. Kev tshawb fawb txhawb nqa:
Kev Sab Laj: Muab cov kev taw qhia ntawm cov txheej txheem compound ntawm kev ua thiab cov ntawv thov.
Kev tsim qauv tsim: Pab cov neeg siv tshawb fawb hauv kev tsim cov txheej txheem sim.
Kev txhais cov ntaub ntawv: Muab kev txhawb nqa rau kev txhais cov ntaub ntawv tshawb fawb.
2. Cov Lus Qhia Zoo:
Cov Ntaub Ntawv Zoo: Muab pov thawj cov ncauj lus kom ntxaws ntawm kev tsom xam (COA).
Cov ntaub ntawv ruaj khov: Muab kev nrawm thiab ntev - dua cov ntaub ntawv kawm ruaj khov kawm cov ntaub ntawv.
Cov Kev Pabcuam Customizization: Peb muab cov kev pabcuam customization rau cov kev sib txawv thiab ntim khoom sib txawv.
3. Kev xa khoom thoob ntiaj teb:
Kev thauj mus los txias: Kub {- tswj kev thauj mus thoob txhua txoj kev kom ntseeg tau tias cov khoom ruaj khov.
Cov Ntawv Txhawb: Muab cov ntawv xa mus ua tiav thiab cov kev lis kev cai ua kom meej cov ntaub ntawv.
Cov lus teb ceev: Teb rau cov neeg siv khoom lus nug thiab xaj hauv 24 teev.
Vim li cas thiaj xaiv Hepius hom GW501516?
TxawvLub tshuab: Ib tug xaiv heev pppp - Δ agonist nrog ib qho kev ua kom meej meej ntawm kev nqis tes ua.
Nyiaj tauYam ua kom zoo dua: Tseem ceeb txhim kho Aerobic endurance thiab kev ua kis las
Txhim khometabolism: Txhim kho cov ntshav lipid profile thiab insulin rhiab
Zoo dua qub: Raw Khoom Siv Purity ntau dua los yog sib npaug rau 99.5%, nruj me ntsis tswj
Lub ntsiab
Hepius hom gw 501516 10 mg ntsiav tshuajsawv cev rau lub tswv yim ntawm metabolic modulator tshawb fawbCov. DhauKev tswj hwm nruj heev, tsim kev tsim tawm kev txhawb nqa thev naus laus zis, thiab cov kev tshawb fawb kev txhawb nqa,Nws muabhigh - Cov Cuab Yeej Zoo Thiab Cov Khoom Siv Hluav Taws XobrauKev tshawb fawb kis las thiab cov kev tshawb fawb ntawm tus kab mob metabolicCov. Xaiv Hepius txhais tau tias xaivKev Tshawb Fawb - qib ua tau zoo thiab kev paub tseeb.
Xav tau kev tshawb fawb lossis cov kev sib tham ntxiv?
Txais tos hu rau Hepius tshawb fawb pab txhawb pab neeg rau kev pabcuam tshaj lij!
NEED dab tsi, thov hu raupeb
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Cim npe nrov: Hepius GW 501516 10 mg * 100 / lub raj mis slam ntsiav tshuaj, Suav teb cov ntsiav tshuaj ntawm qhov ncauj ntawm cov ntsiav tshuaj ntawm qhov ncauj, cov chaw muag khoom, lub hoobkas

