CJC-1295 (muaj DAC) 2mg / vial core qhia
Pharmaceutical -qib peptide formulations|Ntev-kev loj hlob hormone- tso tawm cov tshuaj hormone analogue ua nyob rau hauv Suav teb, 2mg / vial
Specifications2mg / lub raj mis, 10 fwj / lub thawv
Purity: Ntau dua lossis sib npaug li 99% (HPLC kuaj pom)
Qhov tshwm sim: Dawb lyophilized hmoov
Cia: Txias ntawm 2-8 degree, tiv thaiv los ntawm lub teeb. Siv tam sim ntawd tom qab reconstitution.
Core zoo thiab muaj nuj nqi
CJC-1295 (muaj DAC) yog antev -kev loj hlob hormone- tso tawm cov tshuaj hormone analog hloov nrog cov tshuaj affinity complex . Nws ua rau lub neej ntev ib nrab -los ntawm reversibly khi rau albumin nyob rau hauv cov ntshav, thiab nws muaj nuj nqis nyob rau hauv cov kev tshawb fawb uastsis tu ncua txhawb kev tso tawm ntawm endogenous loj hlob hormone.
✅ Ntev-kev ua haujlwm ntev:
Kev hloov kho DAC: Cov tshuaj affinity complex reversibly khi rau cov ntshav albumin, tsim ib tug sustained - tso reservoir.
Kev tso tawm tsis tu ncua: Cov peptide nquag tuaj yeem tso tawm tsis tu ncua rau 7-10 hnub tom qab ib koob tshuaj.
Kev kho mob homeostasis: Ua kom ruaj khov ntawm kev loj hlob hormone thiab IGF-1 nyob rau hauv lub cev muaj zog.
Pulse tuav: Thaum tuav lub sijhawm ntev - ua yeeb yam, nws tseem khaws ib feem ntawm pulsatile secretion yam ntxwv ntawm kev loj hlob hormone.
✅Qualityqhov zoo ntawm Suav manufacturers:
Site-kev hloov kho tshwj xeeb: Precise DAC hloov kho tshuab rau lysine residues xyuas kom muaj kev hloov kho zoo ib yam.
Kev ua kom huv huv: Kev sib xyaw ntawm ion txauv thiab hydrophobic chromatography yog siv los tshem tawm peptides tsis hloov.
Kev ua validation: Hauv vitro thiab hauv vivo bioactivity kuaj yog ua ntawm txhua pawg.
Aseptic kev ruaj ntseg: Txias- ziab thiab txhaws tau ua tiav hauv qib B + A ib puag ncig huv.
✅ khoomNta:
Ntev heev ib nrab -lub neej: Cov nyhuv tuaj yeem kav ntev li 7-10 hnub tom qab noj ib zaug.
Kev tswj hwm yooj yim: Tsuas yog 1-2 koob tshuaj ib lub lim tiam yog xav tau, txhim kho kev ua raws.
Stabilization nyhuv: Tsis txhob muaj qhov hloov pauv loj hauv kev loj hlob cov tshuaj hormones.
Kev siv hauv qhov kev tshawb fawb no: Haum rau cov qauv kev tshawb fawb uas xav tau kev loj hlob ntawm cov tshuaj hormone stimulation.
Daim ntawv qhia kev siv thiab khaws cia
1. Kev kho dua tshiab:
Kev xaiv cov kuab tshuaj: Cov dej tsis huv rau kev txhaj tshuaj (cov kab mob endotoxin<0.25 EU/ml) must be used.
Txuj kev npaj: Txhaum 1 ml ntawm cov dej tsis muaj menyuam rau kev txhaj tshuaj rau hauv 2 mg hmoov vial kom tau txais cov tshuaj nrog cov concentration ntawm 2 mg / ml.
Cov txheej txheem dissolving: Maj mam ncuav cov kuab tshuaj raws phab ntsa ntawm lub raj mis, cia nws sawv ntsug li 2-3 feeb, ces maj mam tig kom yaj.
Lus ceeb toom: Tsis txhob siv cov kuab tshuaj uas muaj cov tshuaj tua kab mob, vim qhov no yuav cuam tshuam rau DAC cov yam ntxwv sib txuas.
2. Cia tej yam kev mob:
Tsis qhib: Khaws ntawm 2-8℃mus txog 24 lub hlis. Tsis txhob khov.
Rov tsim dua: Siv tam sim tom qab hloov kho; cia tsis pom zoo.
Kev thauj mus los: Kev thauj mus los ntawm cov saw txias thoob plaws (2-8 degree), siv cov khoom ntim tshwj xeeb txias.
Kev ruaj ntseg: Cov hmoov lyophilized muaj kev ruaj ntseg zoo nyob rau hauv kev cia khoom kom zoo.
3. Txuj kev noj tshuaj:
Txoj kev tswj hwm: Kev txhaj tshuaj subcutaneous tob rau hauv plab, ncej puab, lossis sab caj npab.
Ib koob tshuaj: 1-2 mg rau ib koob (hloov raws li kev tshawb fawb qauv)
Kev siv ntau zaus: 1-2 zaug hauv ib lub lis piam
Lub sijhawm tswj hwm: Nws raug pom zoo kom muab tshuaj rau lub sijhawm teem tseg (xws li, txhua hnub Monday sawv ntxov).
Kev kho mob ntev: Feem ntau 4-8 lub lis piam ntawm kev siv tas li.
4. Cov lus qhia txog kev hloov tshuaj noj:
Pib koob tshuaj: 1 mg ib zaug ib lub lim tiam, soj ntsuam cov lus teb rau 2 lub lis piam.
Kho koob tshuaj: Kho rau 1-2 mg / koob, 1-2 zaug hauv ib lub lis piam, nyob ntawm cov lus teb.
Cov koob tshuaj ntau tshaj: Nws tsis pom zoo kom ntau dua 2 mg rau ib koob, lossis tag nrho cov koob tshuaj txhua lub lim tiam ntau dua 3 mg.
Kev kho tshwj xeeb: Cov laus lossis cov qauv rhiab yuav tsum pib nrog 0.5 mg rau ib koob.
5. Kev kho mob sib xyaw ua ke:
Siv ua ke nrog GHRP:
CJC-1295 DAC: 1 mg, ib zaug lossis ob zaug hauv ib lub lis piam.
GHRP-2/6: 100-200 mcg, 2-3 zaug ib hnub
Qhov zoo: Ntev -cov nyhuv kav ntev + kev ua kom lub cev muaj zog, ua raws li cov qauv kev tso tawm ntawm lub cev.
Lub caij nyoog txheej txheem:
Lub sijhawm thauj khoom: 1 mg, ob zaug hauv ib lub lis piam rau 2 lub lis piam sib law liag
Lub sijhawm tu: 1-1.5 mg ib zaug ib lub lim tiam rau 4-6 lub lis piam.
Lub sijhawm luv luv: Txiav tshuaj rau 2-4 lub lis piam los soj ntsuam cov teebmeem mus sij hawm ntev.
Vim li cas thiaj xaiv Suav - ua CJC-1295 (xws li DAC)?
TechnicalKev txawj ntse: Paub qhov tseeb ntawm DAC qhov chaw- qhia kev hloov kho thiab ua kom huv huv
ruaj khovzoo: Batch-rau-batch hloov kho tus nqi thiab coefficient ntawm variation ntawm kev ua<5%
Nqi-kev ua tau zoo: Loj- nplai ntau lawm muab cov nqi sib tw thoob ntiaj teb
TechnicalKev pabcuam: Muab cov ntaub ntawv qhia ntxaws ntxaws thiab kev daws teeb meem tsim kev txhawb nqa.
ntseeg tausaw hlau: ib qho kev tswj xyuas zoo los ntawm cov khoom siv raw mus rau cov khoom tiav
Tshawb nrhiav thiab siv cov lus qhia
Ntev - kev tshawb fawb cuam tshuam:
Lub sij hawm ntev - cuam tshuam ntawm kev loj hlob tsis tu ncua cov tshuaj stimulation ntawm cov metabolism
Kev tshawb fawb sib piv ntawm kev loj hlob hormone mem tes thiab cov qauv tso tawm tsis tu ncua
Pharmacokinetic thiab pharmacodynamic yam ntxwv ntawm DAC- hloov peptides
Preclinical kev tshawb fawb:
Tshawb nrhiav lwm txoj kev kho mob rau kev loj hlob hormone deficiency
Kev tshawb fawb txog kev txhawb nqa metabolic rau cov kab mob nkim ntev
Kev cuam tshuam kev tshawb fawb ntawm sarcopenia thiab frailty
Mechanism ntawm kev kawm ua:
Cov kev hloov pauv hauv cov kev taw qhia qis qis vim qhov ua rau GHRH receptor ua kom tsis tu ncua
Kev yoog raws thiab kev hloov pauv hauv kev loj hlob hormone tawm tswv yim kev tswj hwm txoj cai
Kev faib tawm thiab cov yam ntxwv metabolic ntawm albumin - khi peptides
Cov ntsiab lus
Cov khoom no sawv cevqib siab ntawm kev tshawb fawb thiab kev tsim cov tshuaj ntev -peptide ua yeeb yam hauv Suav teb. Los ntawmadvanced DAC kev hloov kho thev naus laus zis, kev tswj xyuas zoo, thiab kev pabcuam kev tshawb fawb, nws muab cov kws tshawb fawb thoob ntiaj teb nrogsiab - zoo CJC-1295 (muaj DAC) cov cuab yeej peptides. Nwsultra-ntev ib nrab- lub neej thiab kev siv tshuaj yooj yimua nwsib qho kev xaiv zoo tshaj plaws rau kev tshawb fawb xav tau kev loj hlob tsis tu ncua ntawm cov tshuaj hormone stimulation. Xaiv peb cov khoom txhais tau tias tau txaiscov cuab yeej tshawb fawb txhim khu kev qha thiab kev txhawb nqa kev tshaj lij.
Xav taudab tsi, thov hu raupeb
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