YK11 Sarms Ua nyob rau hauv Tuam Tshoj High-purity Raw Powder

YK11 Sarms Ua nyob rau hauv Tuam Tshoj High-purity Raw Powder
Khoom Taw qhia:
YK11 yog ib qho tshiab xaiv androgen receptor modulator (SARM) uas cuam tshuam los ntawm cov kev txwv ntawm cov leeg nqaij loj hlob los ntawm kev ua kom cov androgen receptors thiab inhibiting myostatin. Cov kev tshawb fawb tau pom nws cov txiaj ntsig zoo hauv kev txhawb nqa lub cev lean lub cev nce thiab txhim kho pob txha pob txha pob txha, uas yuav luag tsis muaj kev pheej hmoo ntawm kev hloov tshuaj estrogen. Nws tau pom tias muaj peev xwm kho tau hauv kev tshawb fawb ntawm cov leeg nqaij dystrophy thiab osteoporosis, muab cov kev taw qhia tshiab rau kev tsim cov ntaub so ntswg.
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YK11 Raw Material Powder Core Taw Qhia

Pharmaceutical -qib raw khoom|Ua nyob rau hauv Suav teb YK11 (myostatin inhibitor)

Tshuaj npe: (2S)-3-(4-acetamidophenoxy)-2-hydroxy-2-methyl-N-(4-nitro-3-trifluoromethylphenyl)propionamide

CAS Nr.: 431579-34-9

EINECS ID: 610-711-3

Cov mis mos molecular: C₂₀H₂₀F₃N₃O₅

Molecular hnyav: 439.39

Melting pointKub: 152-155 degree

Qhov tshwm sim: Dawb crystalline hmoov

Purity: Ntau dua lossis sib npaug li 99% (HPLC kuaj pom)


Cov teebmeem tseem ceeb

YK11 yog aXaiv androgen receptor modulator (SARM)uas yog dav siv nyob rau hauvKev tshawb fawb cov leeg nqaij hypertrophy, kev kho mob nqaij atrophy, thiab kev ua kis las ncaws pobvim nwstshwj xeeb myostatin inhibition mechanism thiab ib feem agonist zog.

Dual mechanism ntawm kev ua:

Myostatin inhibition: inhibits myostatin signaling pathway, li no relieving nqaij loj hlob txwv.

Ib nrab agonist: Raws li ib feem agonist ntawm androgen receptors, nws txhawb cov leeg nqaij protein synthesis.

Gene qhia: Upregulation of myogenic regulatory factors (MRFs) qhia

✅Qualityqhov zoo ntawm Suav manufacturing:

Purity Guarantee: Raw khoom purity Ntau dua los yog sib npaug rau 99.5%, ua raws li USP cov qauv.

Chirality tswj: S-configuration optical purity Ntau dua lossis sib npaug li 99.8%

Zoo heev stability: Purity tseem siab dua 97% tom qab 6 lub hlis ntawm kev ntsuas nrawm.

✅ thoob ntiaj tebmuab kev ruaj ntseg:

Cold chain logistics: -20℃txias saw tsheb thauj mus los thoob plaws tag nrho cov txheej txheem los xyuas kom meej cov khoom ruaj khov.

Ntau- khoom xa tuaj: Cov tsev khaws khoom hauv cheeb tsam tau tsim nyob rau hauv Suav teb, Tebchaws Europe, Amelikas, thiab Asia - cheeb tsam Pacific, ua kom cov khoom xa tuaj hauv 7 hnub.

Kev them nyiaj yug kev lis kev cai clearance: Kev npaj cov ntaub ntawv ua kom muaj kev lis kev cai zoo thoob ntiaj teb.


Cov txheej txheem ntau lawm thiab kev ruaj ntseg zoo

1. Advanced synthesis txheej txheem:

Asymmetric synthesis: chiral catalytic synthesis, enantiomeric ntau tshaj los yog sib npaug rau 99.8%

Kev ua kom huv huv: Npaj HPLC purification, gradient elution, sau ntawm lub ntsiab ncov.

Tshuab ziab khaub ncaws: Lub tshuab nqus tsev qis- kub kom qhuav, noo noo cov ntsiab lus tsawg dua lossis sib npaug li 0.5%

2. Cov qauv kev tswj xyuas nruj:

Tshuaj purity:

Cov ntsiab lus tseem ceeb: 99.0% ~ 101.0%

Cov khoom muaj feem xyuam: Ib qho impurity Tsawg dua lossis sib npaug li 0.1%, tag nrho impurities Tsawg dua lossis sib npaug li 0.5%

Residual solvent: Ua raws li ICH Q3C cov qauv

Lub cev muaj zog:

Particle loj faib: D50 50-100μm

Qhov ceev: 0.4-0.6 g / cm³

Solubility: Ua tau raws li cov qauv rau cov khoom xyaw tshuaj nquag.

3. Cov ntaub ntawv ruaj ntseg:

Ntev -lub sij hawm ruaj khov: Khaws ntawm -20℃rau 24 lub hlis, txhua qhov ntsuas tau ua tau raws li qhov xav tau.

Kev ntsuas nrawm: Tom qab khaws cia ntawm 25℃rau 6 lub hlis, purity txo qis dua los yog sib npaug li 2.0%.

Kev thauj mus los ruaj khov: Kev vibration thiab poob kev xeem dhau.


Cov yam ntxwv ntawm daim ntawv thov thiab qhov zoo

1. Cov yam ntxwv ua tau zoo:

Cov leeg nqaij hypertrophy: Qhov tseem ceeb nce tus ntoo khaub lig- ntu ntu ntawm cov leeg nqaij

Txhawb zog: Qhov tseem ceeb nce siab tshaj plaws thiab lub zog tawg.

Accelerated Rov qab: Tshaj tawm- kev cob qhia rov qab nrawm nrawm dua.

2. Cov yam ntxwv tseem ceeb thiab qhov zoo:

Dual mechanism: Myostatin inhibition + ib nrab androgen receptor agonism

Cov ntaub so ntswg selectivity: Cov leeg nqaij selectivity yog siab dua li cov tshuaj steroids

Cov kev mob tshwm sim tsawg: Tsawg kev pheej hmoo ntawm androgen{0}} cuam tshuam txog kev mob tshwm sim

3. Qhov zoo ntawm kev siv:

Siv tau qhov ncauj: Siab qhov ncauj bioavailability thiab yooj yim rau siv.

Nruab nrab ib nrab -lub neej: Ib nrab-lub neej yog 12-24 teev, haum rau kev noj ib zaug ib hnub.

Cov ntawv thov tshawb fawb: Cov cuab yeej zoo tshaj plaws rau kev tshawb fawb hauv cov leeg nqaij dystrophy thiab cov tshuaj kis las.


Vim li cas thiaj xaiv YK11, ua hauv Suav teb?

Tsim tshiabMechanism: Thawj SARM-zoo li Myostatin Inhibitor

Chiralkev huv: S-configuration optical purity Ntau dua lossis sib npaug li 99.8%

Tshwj xeebkev huv: Tshaj 99% siab purity, nrog kev tswj xyuas nruj.

ruaj khovmuab: Ib qho kev xa khoom tiav ua kom muaj kev xa khoom raws sij hawm thiab txhim khu kev qha.


Cov ntsiab lus

YK11 raw khoom hmoov, ua nyob rau hauv Suav teb,sawv cev rau qib siab - qauv zoo rau cov leeg nqaij hypertrophy tshiab. Los ntawmadvanced chiral synthesis thev naus laus zis, kev tswj xyuas zoo, thiab cov khoom siv ruaj khov,nws muabsiab -cov cuab yeej tshawb fawb zoo heevraukev tshawb fawb thoob ntiaj teb hauv cov kab mob nqaij thiab cov tshuaj kis las. Xaiv "Made in China" txhais tau tias xaivkev tshawb fawb-qib zoo thiab txhim khu kev qha.


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