Hauj lwm lawm

Kev tsis

Rad -150 99}% raw khoom hmoov txheem taw tes

Kws Tshuaj Kho Mob - qib qib raw|Ua hauv Suav teb Rad-150 (TXL-150)

Tshuaj lom neeg npe: Propyl 2-chloro-4 - [(1R, 2s) -1- (2-chloroethyl) aminophlyl) carbamate

Cas tsis muaj.: 1182367-72-1

Molecular Cov Qauv: C₁₄heccl₂n₂o₂

Molecular hnyav: 309.22

Einecs ID: Tseem tos

Melting taw tes: 186-189 degree

Kev tshwm sim: Cov hmoov dawb dawb

Kev coj dawb huv: Ntau dua los yog sib npaug rau 99% (hplc Nrhiav tau)

So: Yooj yim soluble hauv dmo, me ntsis soluble hauv ethanol

Tub ntxhais muaj nuj nqi|Cov teebmeem tseem ceeb

Rad-150 yog aPhau Ntawv Tshiab, Muaj Peev Xwm, Androgen Receptor Modulator (Sarm)uas tau siv dav rauKev kho mob ntawm cov leeg leeg Atrophy, Osteoporosis kev tshawb fawb, thiab kev ua kom lub cevVim nwsKev Tsim Kho Dichlorophenyyl thiab zoo tshaj qhov ncauj Bioavailability.

Xab tawsXaiv Teeb Tshuab:

Siab receptor affinity: Muaj zog androgen receptor binding affinity, EC50 <1 NM

Nqaij Nqaij Xaiv: Xaiv cov kev ua ub no hauv cov leeg thiab pob txha pob txha

Zoo heev rau qhov ncaujuse: oral bioavailability >80%, ntev ib nrab ib nrab - lub neej

Sib thamQhov Zoo Ntawm Suav Raug:

Ultra - purity siab: Cov khoom siv raw ntau dua los yog sib npaug rau 99%, ib qho impurities tsawg dua los yog sib npaug 0.1%

Chiral purity: Kev Purity Optical ntawm Chiral Chaw Loj dua los yog sib npaug rau 99.8%

Crystal Foos Ruaj Khwv: Ib qho ruaj khov - Crystal daim ntawv ua kom muaj cov qauv luam ntawv.

✅globalmuab kev lees paub:

Cov Khoom Siv Txias Txias: Qhov ntsuas kub tas li rau thaum 15-25℃kom ntseeg tau tias muaj peev xwm ruaj khov.

Ntau yam kev xaiv ntim ntim ntim: 1kg / hnab, 5kg / nruas, thiab lwm yam.

Txhawb Nqa Kev Pab Cuam Kev Lis Haujlwm: Ua tiav cov ntaub ntawv xa tawm xws li MSDS thiab COA

Cov Txheej Txheem Ntau Lawm thiab Kev Ntsuas Zoo

1. Qhov zoo ntawm cov txheej txheem synthesis:

Chairal Synthesis: Asymmetric synthisis ua kom ntseeg tau tias kho cov chaw teeb tsa chiral.

Tus Txheej Txheem Purification: Kem chromatography ua ke nrog recrystallization kom tau siab - purity qustals.

Kom Qhuav Tshuab: Lub Tshuab nqus tsev qis -}} pa taws txias, noo noo cov ntsiab lus tsawg dua lossis sib npaug rau 0.5%

2. Nruj metric qauv tswj hwm:

Tshuaj lom neeg purity:

Cov ntsiab lus tseem ceeb: 99.0% ~ 10.0.0%

Related tshuaj: ib leeg tsis paub tsis muaj zog tsawg dua los yog sib npaug rau 0.1%, tag nrho cov impurities tsawg dua los yog sib npaug rau 0.5%

Residual cov kuab tshuaj: ua raws li Ich Q3C qauv

Cov Khoom Siv Lub Cev:

Particle loj faib: d 50 50-100 μm

Bulk ntom: 0.4-0.6 g / cm³

Solubility: ua tau raws cov qauv rau cov khoom muaj cov tshuaj muaj zog.

3. Cov ntaub ntawv ruaj khov:

Ntev -} lub sij hawm ruaj khov: Ruaj khov rau 36 lub hlis ntawm 25℃/ 60% rh.

Nrig kuaj ntsuas: Dhau tom qab 6 lub hlis ntawm 40 Degree / 75% Rh.

Kev thauj mus los ruaj khov: Kev co thiab poob kev sim dhau.

Kev Tshawb Fawb Kev Tshawb Fawb thiab Kev Tshawb Xyuas Kev Tshawb Fawb

1. Kev tshawb fawb thiab cov chaw thov:

Kev kho mob rau cov leeg atrophy: Cancer Cachexia, Hnub Nyoog -} ity ntsig txog sarcopenia

Osteoporosis: Ua kom muaj cov pob txha ceev thiab txhim kho pob txha zoo

Txhim kho lub cev: Cov leeg mob loj thiab lub zog hauv cov neeg ncaws pob

2. Cov ntaub ntawv preclinical:

Khaus cov leeg nce: Cov kev tshawb fawb tsiaj qhia tau 15-20% nce rau hauv cov nqaij ntshiv cev.

Mob pob txha: Tseem ceeb dua cov pob txha ntxhia ntxhia thiab txhim kho pob txha biomechanical cov khoom

Siab Xaiv: Tsawg heev cuam tshuam rau ntawm lub prostate, tus neeg xaiv cov nqaij tseem ceeb.

3. Cov yam ntxwv tseem ceeb thiab cov txiaj ntsig:

Ua tau zoo rau kev tswj hwm qhov ncauj: Nws muaj lub qhov ncauj ntawm qhov ncauj thiab haum rau ntev - lub sij hawm siv.

Ntev ib nrab ib nrab - lub neej: tshem tawm ib nrab - lub neej 24-36 teev, ib zaug noj tshuaj txhua hnub

PunaceSutic qhov rai: Kev Nyab Xeeb Kev Nyab Xeeb, Kev Pheej Hmoo qis ntawm cov kev mob tshwm sim

Kev xa khoom hauv ntiaj teb thiab kev pabcuam kev pabcuam

1. Ntau Lawm Muaj Peev Xwm:

Muaj Peev Xwm Ntau Lawm: Dhau 100 kg ib xyoo

Saj zawg zog tsim: Customized specifications thiab ntim khoom yuav tsum tau.

Muaj Peev Xwm Muaj Peev Xwm Muaj Peev Xwm: Ntau cov kab ntau lawm ua kom tau cov khoom ruaj khov

2. Ntawv pov thawj zoo:

Daim Ntawv Pov Thawj Ntawv Pov Thawj: Muaj ntawv pov thawj los ntawm ISO 9001 Kev Tswj Xyuas Kev Tswj Xyuas Zoo

Ua raws li cov qauv: Raws li cov qauv khoom siv raw tshuaj

Ua tiav Cov Ntaub Ntawv: Muab cov pob ua tiav cov ntaub ntawv zoo.

Vim li cas thiaj xaiv Suav - ua rad-150?

Heevxaiv: Muaj kev sib luag rau cov khoom lag luam Androgen, EC50 <1 nm

Txaus qhuaskev coj dawb huv: Hla 99% siab purity, nrog tswj kev tswj nruj.

Tau siab kawgtej txuj ci tshiab: Cov txheej txheem chairal, kev ua kom zoo nkauj txog li 99.8%

Vam taumov: Loj - nplai ntau lawm muaj peev xwm, xa sijhawm

Lub ntsiab

Rad -150 99} kev ntshiab raw hmoov hmoov, ua nyob rau hauv Suav teb,sawv cev qhov siab - zoo qauv ntawm kev muaj zog thiab xaiv Androgen Revenor ModulatorCov. DhauAdvanced Chiral synthesis, kev tswj hwm nruj heev, thiab lub zog ruaj khov, nws muabhigh - Zoo, heev nquag tshawb cov ntaub ntawv raw rau cov kev tshawb fawb thoob ntiaj teb ntawm cov leeg atrophy thiab osteoporosisCov. Xaiv ua nyob rau hauv Suav teb txhais tau tias xaivKev Zoo Tshaj Plaws thiab Kev Ruaj Ntseg Txhawb.

Xav tau cov qauv lossis cov ntaub ntawv ua haujlwm?

Xav tiv tauj peb cov pab thiab pab neeg ua haujlwm rau kev ua haujlwm!

Xav taudab tsi, thov hu raupeb