1. Basic Chemical & Physical Properties
|
Yam khoom |
Parameter |
|---|---|
|
CAS Nr |
54965-24-1 |
|
EINECS Number |
259-410-8 |
|
Molecular Formula |
C₃₂H₃₇NO·C₆H₈O₇ |
|
Molecular Luj |
563.64 |
|
Melting Point |
140℃- 142 degree |
|
Qhov tshwm sim |
Dawb crystalline hmoov |
2. Kev siv dav dav
Tamoxifen Citrate (Nolvadex) yog ib qho tseem ceeb xaiv Estrogen Receptor Modulator (SERM), dav siv los ntawm bodybuilders rau Post-Cycle Therapy (PCT). Nws ua hauj lwm pab raws li ib qho tseem ceeb auxiliary compound rau steroid cycles, zoo inhibiting estrogenic phiv thiab restores ntuj hormonal theem. Yuav luag txhua tus neeg ncaws pob sib tw suav nrog Nolvadex rau hauv lawv lub voj voog thiab tom qab- cov txheej txheem voj voog kom ruaj ntseg tau txais kev cob qhia thiab tswj lub cev ruaj khov.
3. Cov yam ntxwv ntawm cov khoom
Nolvadex yog qhov ncauj formulation ntawm Tamoxifen, featuring tshwj xeeb xaiv estrogen receptor modulation zog. Nws ua raws li estrogen antagonist nyob rau hauv cov ntaub so ntswg ntawm lub mis thaum ua hauj lwm raws li ib tug estrogen agonist nyob rau hauv lwm yam ntaub so ntswg ntawm lub cev. Nws precisely thaiv cov tshuaj estrogen receptors hauv zos los tiv thaiv gynecomastia thiab cov dej tuav ntau dhau, tsis muaj kev cuam tshuam tag nrho cov tshuaj estrogen.
Sib txawv los ntawm hnyav Aromatase Inhibitors (AIs), Tamoxifen khaws cov txiaj ntsig zoo ntawm lub cev ntawm cov tshuaj estrogen rau kev noj qab haus huv ntawm cov hlab plawv thiab cov pob txha ntom ntom, xa cov kev tswj hwm hormonal zoo dua. Nrog rau qhov zoo ntawm qhov ncauj bioavailability thiab pib sai, nws tuaj yeem txo qhov tsis xis nyob thaum ntxov estrogenic xws li txiv mis rhiab heev thaum lub voj voog.
Raws li ib tug tseem ceeb PCT compound, Nolvadex zoo reactivates Hypothalamic{0}}Pituitary-Testes-Axis (HPTA). Nws txhawb nqa kev tso tawm ntawm Luteinizing Hormone (LH) thiab Follicle-Stimulating Hormone (FSH), sai sai rov pib endogenous testosterone ntau lawm, uas yog ib qho tseem ceeb rau tom qab- lub voj voog rov qab thiab cov leeg nqaij tuav.
4. Cov khoom siv tseem ceeb
4.1 Gynecomastia Tiv Thaiv & Tshaj Tawm -Cycle Hormone Recovery
Tamoxifen Citrate occupies estrogen receptors nyob rau hauv lub mis cov ntaub so ntswg, fundamentally tiv thaiv thiab inhibiting txiv neej gynecomastia txoj kev loj hlob. Hauv cov txheej txheem PCT cov txheej txheem, nws ua kom rov qab los ntawm endogenous testosterone tom qab siv exogenous steroid. Nws pab cov neeg siv khaws cov leeg nqaij ntshiv, zam kom tsis txhob muaj rog rog, thiab ua kom lub siab thiab libido, kom ntseeg tau tias du thiab nyab xeeb tom qab- rov qab mus.
4.2 Lipid Txoj Cai & Kev Tiv Thaiv Pob Txha
Tamoxifen muab kev tswj hwm tshuaj estrogen me me thiab tsis muaj kev phiv hnyav tshwm sim los ntawm cov tshuaj aromatase inhibitors. Nws ua kom zoo dua HDL-LDL cov roj cholesterol piv, muaj txiaj ntsig offsetting lipid siab coj los ntawm qhov ncauj steroids. Lub caij no, nws tswj cov pob txha pob txha pob txha pob txha los ntawm kev khaws cov tshuaj estrogen cov pob txha- tiv thaiv kev ua haujlwm, ua rau nws muaj kev ntseeg siab ntev ntev - cov tshuaj hormonal tswj kev daws teeb meem rau cov neeg siv zog.
5. Cov ntaub ntawv tiv tauj
Rau cov khoom nug, kev txiav txim ntau thiab kev txhawb nqa, thov hu rau peb:
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