Finasteride (Finasteride) Raw Khoom Hmoov Core Taw Qhia
Kws Tshuaj Ua Lag Luam Qib Khoom Qhua Khoom xyaw|Cov ({5 -} reductase inhibitor)
Tshuaj lom neeg npe: N {- tert - butyl-3-}} {}} carboxamide
Tus lej: 98319-26-7
Einecs tooj: 619-695-6
Molecular Cov Lus: C₂₃h₃₆n₂o₂
Molecular hnyav: 372.55
Melting taw tes: 252-254 degree
Zog: Dawb lossis tawm -} e} crystalline hmoov
Solubility: me ntsis soluble hauv dej, yooj yim soluble hauv methanol thiab ethanol
Cov khoom tseem ceeb
Finasteride yog aHom II {5 -} reductase inhibitoruasinhibits qhov hloov dua siab tshiab ntawm testosterone rau dihydotestosterone (DHT)thiab tau siv davHauv kev kho mob androgenic alopecia thiab benign prostatic hyperplasia.
✅ Pharmacological cov zog:
Cov Inhibition heev Inhibition: Kev tiv thaiv Inhibitory kev ua txhaum tawm tsam hom II 5 -} reductase yog 100 npaug siab dua qhov uas tawm tsam hom i
DHT txo: Ib qho dej ntawm ib qho ntawm qhov ncauj tuaj yeem txo cov ntshav dej DHT qib los ntawm 70%
Cov nqaij tshwj xeeb: feem ntau cuam tshuam tus prostate thiab cov tawv taub hau
✅ Kev Nyab Xeeb Nta:
Siab Xaiv: tsis cuam tshuam rau cov synthesis ntawm lwm cov tshuaj steroid
Zoo zam: Cov kev mob tshwm sim tau mob me thiab thim rov qab hauv feem ntau cov neeg mob
Ntev - sij hawm kev nyab xeeb: Ntau tshaj 20 xyoo siv thiab cov ntaub ntawv muaj kev nyab xeeb txaus
Muaj peev xwm kawg cov khoom lag luam thiab cov ntawv thov
1. Daim duab Ntsej Muag (1mg / 5mg):
Txoj Kev Tsim:
Cov Khoom Siv Ru Khoom Siv: 1Mg lossis 5MG
Microcrystalline Cellulose: Muab Tub Ntxaij
Croscarmellose sodium: tsis sib tua
Magnesium Stearate: Roj nplua nyeem
Cov Ntawv Thov Kev Kho Mob:
Kev Kho Plaub Hau: 1 mg / hnub rau txiv neej Androgenic alopecia
BPH: 5mg / hnub rau kev kho mob ntawm benign prostatic hyperplasia
Yuav Tsum Tau Txais: Siv tas mus li rau 3-6 lub hlis kom pom cov txiaj ntsig tseem ceeb
2. Kev daws teeb meem (0.1% -0.25%):
Txoj Kev Tsim:
Cov Khoom Siv Ribasteride: 0.1% -0.25%
Ethanol: Hnyav
Propylene Glycol: Nkag Mus Rau Enhancer
Menthol: txias tus neeg sawv cev
Cov Ntawv Thov Kev Kho Mob:
Kev Kho Mob Topic: Thov ncaj qha rau saum tawv taub hau ntawm thaj tsam ntawm cov plaub hau poob
Txo qhov teeb meem raug: Txo kev pheej hmoo ntawm cov kev phiv
Kev Kho Mob: Tuaj yeem siv nrog cov ntsiab lus npaj xws li Minoxidil
3. Microedle hloov chaw:
Txoj Kev Tsim:
Cov Khoom Siv Ru Khoom Siv: 0.05% -0.1%
Hyaluronic Acid: Matrix
Microneedle Array: 500-1000 μm nyob rau hauv ntev
Cov Ntawv Thov Kev Kho Mob:
Kev xa tshuaj TransdleMal: Txhim Kho Cov tawv nqaij nqus daim tawv nqaij nqus los ntawm microedles
Txhim Kho Bioavailability: Zam kev ua ntej -} dhau cov nyhuv
Kev Tso Tawm Tso Tawm: Muab cov lus ntev - sij hawm thiab ruaj khov yeeb tshuaj
4. Compound Cov Plaub Hau Loj Hlob:
Kev sib xyaw ua ke:
Finasteride + minoxidil: Dual kev nqis tes los txhawb cov plaub hau kev loj hlob
Finasteride + biotin: Cov as -fement cov as-ham yuav tsum muaj rau cov plaub hau loj hlob
Finasteride + caffeine: Stimulates plaub hau
Cov kev siv raws tu qauv
1. Dosage Regimen:
Androgenetic alopecia:
Pom zoo koob: 1 mg / hnub, hais lus
Lub sijhawm siv: tsawg kawg 3 lub hlis ntawm kev siv tas mus li
Cov txiaj ntsig zoo tshaj plaws: lub txiaj ntsig tau ua tiav tom qab 12 lub hlis ntawm kev siv
Benign prostatic hyperplasia:
Pom zoo koob tshuaj: 5 mg / hnub, hais lus
Pib pib lub sijhawm: prostate ntim yog txo qis tom qab 6 lub hlis ntawm kev kho mob
Ntev - siv siv: siv tau siv ntau xyoo
2. Kev Siv:
Thawj coj:
Noj ntawm lub sijhawm ruaj khov, ib zaug ib hnub
Tuaj yeem nqa nrog lossis tsis muaj zaub mov
Yuav tsum tau siv txuas ntxiv tsis muaj kev cuam tshuam
Kev coj ntawm kev tswj hwm:
Thov 1-2 zaug ib hnub kom qhuav tawv taub hau
Zaws kom txog thaum nqus tag nrho
Ntxuav tes kom huv si tom qab siv
3. Siv cov neeg tshwj xeeb:
Kev noj tshuaj rau cov laus:
Tsis Muaj Kev Kho Mob
Saib xyuas cov prostate -}} Cov Lus Qhia A Antigen (Psa) Qib
Hepatic tsis txaus:
Mob me rau kev raug mob me me: siv nrog kev ceev faj thiab xav tau kev saib xyuas ze
Kev raug mob hnyav: tsis pom zoo
4. Kev tswj hwm kev tiv thaiv:
Cov kev mob tshwm sim ntau:
Kev Ua Haujlwm Kev Ua Kom Zoo: Kev poob qis Libido, erectile kawg (incidence 1% -3%)
Lwm yam teebmeem: Kev siv lub mis, tawm pob, thiab lwm yam.
Kev Ntsuas Ze:
Feem ntau cov kev mob tshwm sim ploj ntawm lawv tus kheej thaum lub sijhawm noj tshuaj txuas ntxiv.
Yog cov tsos mob pheej yuav tsum tau txiav txim siab lossis txo cov koob tshuaj
Cov kev mob tshwm sim feem ntau yog reversible tom qab nres cov tshuaj
Vim li cas thiaj xaiv cov khoom siv buasteride?
Pov thawj nyhuv: Tshuaj tiv thaiv kev ua pov thawj kom ua tau zoo rau androgenic alopecia
Ntau cov ntaub ntawv ntau npaum: Tuaj yeem npaj tau hauv ntau cov ntawv ntau npaum li cas xws li qhov ncauj thiab tshuaj pleev
Kev Ua Lag Luam Loj Hlob: Thov kom muaj kev kho plaub hau ntxiv kom loj tuaj
Zoo ruaj khov: Cov ntaub ntawv raw yooj yim khaws thiab cov txheej txheem
Tag
Cov ntaub ntawv raw yogCov khoom xyaw tseem ceeb rau kev npaj cov plaub hau kev kho mobCov. DhauCov txheej txheem tsim qauv sib txawv,Lawv tuaj yeem tsim mus rau ntau cov khoom lag luam xaus, suav nrogCov ntsiav tshuaj ntawm qhov ncauj, cov kev daws teeb meem, thiab cov khoom hloov tshiab transdermalCov. Xaiv peb yuav muab rau kojsiab -} Purity raw cov ntaub ntawv, kev txhawb nqa kev ua haujlwm, thiab muaj txhij txhua {{1} kev pab muag khoom.
Xav tau cov txuj ci tshwj xeeb lossis kev qhia txuj ci?
Txais tos tiv toj rau peb cov kws pab txhawb nqa los muab cov kev daws teeb meem!
Xav taudab tsi, thov hu raupeb
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Ntawv xov |
Tag nrho |
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