Kws zoo tshaj plaws cov khoom lus qhia
Cov khoom siv ntshiab cov khoom siv hmoov|Cov tsos ntxwv Aromatase inhibitor raw khoom
Cas tsis muaj.: 107868-30-4
Einecs tooj: 601-818-9
Molecular Cov Qauv: C₂₀h₂₄o₂
Molecular hnyav: 296.41
Melting Taw tes: 191 Qib -195 Degree
Zog: Dawb lossis tawm -} e} crystalline hmoov
Exemestane siv
Exemestane yog ibTsis pub lwm tus neeg InromalleCov. Vim nwsLub zog tshuaj estrogen - suppressing cuam tshuam thiab nws cov xwm txheej uas yog kev kho mob cancer mis, nws yog dav sivHauv kev kho mob cancer mis, estrogen tswj thaum lub sijhawm tshuaj steroid, thiab hauv kev npaj rau kev sib tw ntawm kev sib tw ua haujlwm.
✅ Muaj pes muaj zog tshuaj estrogen:
Irreversibly inhibits aromatase, txo cov qib tshuaj estrogen hauv lub cev los ntawm ntau dua 95%
Ua kom tiav cov kev hloov pauv ntawm testosterone rau estrogen, tshem tawm txoj kev pheej hmoo ntawm cov tshuaj estrogenization thiab dej thiab sodium khaws cia
✅ Kev Kho Mob Cancer Mis:
Thawj - txoj kab adjuvant txoj kev kho rau qhov postperativeEstrogen receptor -}} zoo cancer mis
Ua kom me duaTxoj kev pheej hmoo mob cancer mislos ntawm ntau tshaj 40%
✅ Qoj Apps:
Tiv thaiv kev estrogen -}} cov kev mob tshwm simThaum lub sijhawm sloid voj voog
Tshem tawm cov dej seemthiab txhim kho cov leeg cov leeg thaum npaj kev npaj
Cov yam ntxwv exemestane
Qhov ncauj muaj txiaj ntsig:
Siab qhov ncauj bioavailability(>90%)
Siv ib zaug ib hnub, tsis muaj kev txhaj tshuaj yuav tsum tau
Irrreersible inhibition:
Kev khi mus tas li, xav tau tos kom muaj enzyme tshiab los ua (4-7 hnub)
Cov nyhuv yog ntev -} kav, thiab nws siv sijhawm los rov tsim cov qib estrogen tom qab nres cov tshuaj
Steroid Qauv Zoo:
Tsis muaj Estrogen fougback cuam tshuam ntawm nonsteroidal ais(xws li, letrozole)
Tsawg dua qhov cuam tshuam ntawm cov ntshav khib nyiabthiab cov kev nyab xeeb ntau dua
Nruab nrab ib nrab - lub neej:
24 -} teev ib nrab-lub neej, haum rau ib zaug -} noj su txhua hnub
{-}} Lub xeev cov ntshav ntau dua7-10 hnubmus cuag
Cov ntawv thov EXEMESTANESTANES
Kev Kho Mob Cancer Mis:
Koob Tshuaj Kho Mob: 25mg / hnub x 5 xyoos
Cov hauj lwm zoo: ER + Kev Them Nyiaj Kho Mob Cancer mis> 90%
Cyclic Estrogen tswj:
Tiv thaiv kev txhaj tshuaj: 12.5 mg Txhua Txhua Hnub
Kho cov koob tshuaj: 25 mg / hnub (thaum cov tsos mob ntawm feminization tshwm sim)
Kev sib tw sib tw:
4 lub lis piam ua ntej kev sib tw: 25 mg / hnub → 12,5 mg / hnub (lub lim tiam dhau los)
Cov nyhuv: cov leeg nqaij tawv tawv tawv + xoom subcutous noo noo
EXEMEXE ceev faj
Tsawg estrogen: Tej zaum yuav ua rau mob sib koom tes thiab txha caj qaum (calsteoporosis (calsteoporosis (calcium / vitamin D ntxiv ntxiv yuav tsum tau)
Ntshav lipid soj ntsuam: Ntev {- siv tau tej zaum yuav cuam tshuam rau cov ntshav lipid lipid (cov tshev yuav pom zoo)
Cov poj niam cev xeeb tub yog txwv tsis pub siv cov khoom no: Nws yuav ua rau menyuam pw tsis zoo (cov poj niam ntawm lub hnub nyoog menyuam yaus yuav tsum nruj me ntsis ua raws li Kev Tiv Thaiv Kev Tiv Thaiv)
Vim li cas thiaj xaiv Exemestane?
Ib qho ntawmCov feem ntau muaj prolomatase inhibitors, nrog kev tsis paub tab thiab ntev -} kav ntev ntawm inhibitos cuam tshuam
Tus qauv kub rau kev kho mob cancer mis, nws txoj kev nyab xeeb tau nthuav dav kev kuaj xyuas
Qhov kawg xaiv rau kev sib tw npaj, kiag li tshem tawm kev ntxhib los ua kom tiav "qhuav thiab nyuaj" xeev
Kev Muaj Peev Xwm Zoo:
GMP -} ua tiav ntau lawm, txhua pobHPLC Purity kuaj (loj dua lossis sib npaug rau 99%
Thib peb - tog kab ke ceeb toom (COA)suav nrog cov khoom
Lub Ntiaj Teb Shipping:
Thawj Ntim Ntim Ntim, ntiag tug xa
Tag
Exemestane yogLub zog tshaj plaws rau estrogen tswj, tshwj xeeb haum rauKev kho mob cancer mis, siab-}} Kev npaj steroid mus, thiab npaj kev sib twCov. Cov koob tshuaj pom zoo yog12.5-25mg / hnub.
Xav tau phiaj xwm kho tshuaj tshwj xeeb?
Peb muab cov tshuaj tshaj lij kev tshaj tawm los pab koj ua tiav koj cov hom phiaj nyab xeeb thiab zoo!
Yog tias koj xav tau dab tsi, thov hu rauTag nrho
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Cim npe nrov: Exemasin (Aromasin) 99% Purity Hmoov, Tuam Tshoj Exemasin) 99% Purity Hmoov Manufacturers, lwm tus neeg, Hoobkas

