Aastrozole (ArimideX) 99% hmoov nplej nyoos

Aastrozole (ArimideX) 99% hmoov nplej nyoos
Khoom Taw qhia:
Anastrozole yog lub zog muaj zog procomase inhibitor uas thim rov qab aromatase kev ua si hauv lub cev (los ntawm 70- 80%). Nws yog qhov ua tau zoo hauv kev tswj hwm tus mob cancer mis thiab hauv kev tswj hwm kev tswj hwm cov kev mob tshwm sim (xws li Gynecomastia thiab Edema) thaum lub voj voog tshuaj steroid. Cov tshuaj qis sib txawv (piv txwv li, 0.5 mg / lub lim tiam) tuaj yeem sib npaug ntawm cov kev cuam tshuam ntawm cov kev sib koom tes zoo li muaj zog inhibitors xws li letrozole.
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Hauj lwm lawm
Kev tsis

Aastrozole (Aastrozole) Raw Khoom Hmoov Core Taw Qhia

Kws muag tshuaj -} qib raw cov ntaub ntawv|Aastrozole, ib tug heev xaiv aromatase inhibitor

Tshuaj lom neeg npe: 2,2 '{{- [5,2,4-triazol-1-ylmethyl) -1,3-phenyfene] BIS (2-Methylpropionitrile)

Tus lej: 120511-73-1

Molecular cov mis: c₁₇h₁₉n₅

Molecular hnyav: 293.37

Melting Taw tes: 81-85 Degree

Zog: Dawb lossis tawm -} e} crystalline hmoov

Purity: ntau dua los yog sib npaug rau 98% (HPLC)


Cov teebmeem tseem ceeb

Anastrozole yog aSiab heev xaiv nonsteroidal aromatase inhibitorCov. Vim nwsMuaj Peev Xwm Estrogen - suppressing cov khoom thiab kev tsim txom zoo, nws yog dav sivHauv kev kho mob cancer mis, kev tiv thaiv ntawm estrogen -}} kev phiv, thiab cov tshuaj estrogen thaum lub sij hawm steroid.

Muaj pes muaj zog tshuaj estrogen:

Thim rov qab los ntawm aromatase, inhibiting qhov hloov dua siab tshiab ntawm androgens rau estrogens

Txo cov qib estradiollos ntawm ntau tshaj 85%, tswj tau zoo tshuaj estrogen -}} cov kev mob tshwm sim

Siab Xaiv Tau Zoo:

Tshwj xeeb inhibits aromatasetsis cuam tshuam rau cov synthesis ntawm lwm cov tshuaj steroid

Tsis cuam tshuam nrog adrenal cortical hormones synthesis, muaj kev nyab xeeb dua

Daim Ntawv Thov Kev Kho Mob Cancer mis:

Kev kho mob ntawm postmenopausal lub mis cancer, zoo inhibiting cov qog kev loj hlob

Zoo zamthiab muaj kev nyab xeeb rau ntev - tsis siv

Qhov Zoo:

Siab qhov ncauj bioavailability(83%) thiab siv tau yooj yim

Ntev ib nrab ib nrab - lub neej(50 teev), tso cai rau ib zaug -} noj txhua hnub

Zoo zam nrogTsawg txoj kev pheej hmoo ntawm cov kev mob tshwm sim


Kawg Cov Khoom Qhia Khoom Siv Khoom Taw Qhia

1. Tablet npaj (1 mg / ntsiav tshuaj):

Piv Txwv Piv Txwv(rau 1000 ntsiav tshuaj):

Anastrozole Raw Khoom: 1.0G

Microcrystalline Cellulose: 80.0g

Lactose: 50.0g

Hla -} Txuas cov carboxymethyl cellulose sidium: 8.0g

Magnesium Stearate: 2.0g

Npaj txheej txheem:

Cov Khoom Siv Raw Ua Ntej: Micronization (D90 tsawg dua los yog sib npaug rau 10μm)

Cov nqi sib xyaw sib xyaw: maj mam sib tov nrog rau dituent

Ntub av granulle: Granulate nrog cov nyiaj uas tsim nyog ntawm cov dej huv thiab qhuav hauv cov kua hauv 50 degree

Granulation: 20 Mesh Sab Canules, ntxiv Flow AIDS thiab roj nplua nyeem

Ntsiav tshuaj: 6 hli round tuag, 8-10knights ntsiav tshuaj

Zaj duab xis txheej: Gastro - soluble zaj duab xis txheej kom txhim kho kev ruaj khov thiab palatability

Kev Tswj Xyuas Zoo:

Cov ntsiab lus sib xyaw: RSD tsawg dua lossis sib npaug ntawm 3% (UV {{1} hplc nrhiav kom pom)

Tus lej sib cais: Ntau dua los yog sib npaug rau 85% hauv 30 feeb (duav txheej txheem, 50 rpm)

Lwm yam tshuaj: Ib leeg impurity tsawg dua los yog sib npaug rau 0.5%, tag nrho cov impurities tsawg dua los yog sib npaug rau 1.0%

2. Npaj sau ntawv:

Cov Khoom Siv Raw Khoom Raw: tsis - steroidal qauv, txom dej solubility

Ib Cheeb Tsam Ntau Lawm: txheeb ze cov av noo tsawg dua los yog sib npaug 40%, noo noo - eam pov thawj kho

Ntim yuav tsum tau: Aluminium ntawv ci tshuab ntim, lub teeb - ntawv pov thawj thiab noo noo-


Vim li cas thiaj xaiv Aastrozole?

Siab xaiv Aromatase inhibitorNrog kev pheej hmoo ntawm cov kev mob tshwm sim

Muaj zog estrogen tswj, txhim khu kev qha nyhuv

Kev thev siab zoothiab muaj kev nyab xeeb rau lub sijhawm ntev - tsis siv


Kev Muaj Peev Xwm Zoo:

GMP -} ua tiav ntau lawm, txhua pobHPLC Purity kuaj (loj dua lossis sib npaug rau 98%)

Thib peb - tog kab ke ceeb toom (COA)suav nrog cov khoom

Microbial txwv kuajTxhawm rau kom muaj kev nyab xeeb

Lub Ntiaj Teb Shipping:

Thawj Ntim Ntim Ntim, noo noo - ntawv pov thawj thiab lub teeb- ntawv pov thawj

Ntiav neeg, tsis muaj logo ntawm lub ntim sab nraud

Kub -} tswj kev thauj mus losTxhawm rau kom muaj kev ruaj khov


Tag

Aastrozole tuaj yeem yogtsim rau hauv kev siv cov tshuaj lim dej siv cov txheej txheem txheemCov. Nws yog tshwj xeeb rauKev kho mob cancer mis, kev tiv thaiv ntawm estrogen -}} kev phiv, thiab cov tshuaj estrogen thaum lub sij hawm steroidCov. Cov koob tshuaj pom zoo yog1 mg / hnub.

Xav tau phiaj xwm npaj phiaj xwm tshwj xeeb?

Peb muab cov kev coj ua kev tshaj lij los pab koj npaj cov khoom kawg kom nyab xeeb thiab zoo!


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Cim npe nrov: Aastrozole (ArimideX) 99% Hmoov Nplej, Tuam Tshoj areask) 99% Cov Khoom Siv Hmoov Nplej, Chaw muag khoom, Hoobkas

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