Aastrozole (Aastrozole) Raw Khoom Hmoov Core Taw Qhia
Kws muag tshuaj -} qib raw cov ntaub ntawv|Aastrozole, ib tug heev xaiv aromatase inhibitor
Tshuaj lom neeg npe: 2,2 '{{- [5,2,4-triazol-1-ylmethyl) -1,3-phenyfene] BIS (2-Methylpropionitrile)
Tus lej: 120511-73-1
Molecular cov mis: c₁₇h₁₉n₅
Molecular hnyav: 293.37
Melting Taw tes: 81-85 Degree
Zog: Dawb lossis tawm -} e} crystalline hmoov
Purity: ntau dua los yog sib npaug rau 98% (HPLC)
Cov teebmeem tseem ceeb
Anastrozole yog aSiab heev xaiv nonsteroidal aromatase inhibitorCov. Vim nwsMuaj Peev Xwm Estrogen - suppressing cov khoom thiab kev tsim txom zoo, nws yog dav sivHauv kev kho mob cancer mis, kev tiv thaiv ntawm estrogen -}} kev phiv, thiab cov tshuaj estrogen thaum lub sij hawm steroid.
✅ Muaj pes muaj zog tshuaj estrogen:
Thim rov qab los ntawm aromatase, inhibiting qhov hloov dua siab tshiab ntawm androgens rau estrogens
Txo cov qib estradiollos ntawm ntau tshaj 85%, tswj tau zoo tshuaj estrogen -}} cov kev mob tshwm sim
✅ Siab Xaiv Tau Zoo:
Tshwj xeeb inhibits aromatasetsis cuam tshuam rau cov synthesis ntawm lwm cov tshuaj steroid
Tsis cuam tshuam nrog adrenal cortical hormones synthesis, muaj kev nyab xeeb dua
✅ Daim Ntawv Thov Kev Kho Mob Cancer mis:
Kev kho mob ntawm postmenopausal lub mis cancer, zoo inhibiting cov qog kev loj hlob
Zoo zamthiab muaj kev nyab xeeb rau ntev - tsis siv
✅ Qhov Zoo:
Siab qhov ncauj bioavailability(83%) thiab siv tau yooj yim
Ntev ib nrab ib nrab - lub neej(50 teev), tso cai rau ib zaug -} noj txhua hnub
Zoo zam nrogTsawg txoj kev pheej hmoo ntawm cov kev mob tshwm sim
Kawg Cov Khoom Qhia Khoom Siv Khoom Taw Qhia
1. Tablet npaj (1 mg / ntsiav tshuaj):
Piv Txwv Piv Txwv(rau 1000 ntsiav tshuaj):
Anastrozole Raw Khoom: 1.0G
Microcrystalline Cellulose: 80.0g
Lactose: 50.0g
Hla -} Txuas cov carboxymethyl cellulose sidium: 8.0g
Magnesium Stearate: 2.0g
Npaj txheej txheem:
Cov Khoom Siv Raw Ua Ntej: Micronization (D90 tsawg dua los yog sib npaug rau 10μm)
Cov nqi sib xyaw sib xyaw: maj mam sib tov nrog rau dituent
Ntub av granulle: Granulate nrog cov nyiaj uas tsim nyog ntawm cov dej huv thiab qhuav hauv cov kua hauv 50 degree
Granulation: 20 Mesh Sab Canules, ntxiv Flow AIDS thiab roj nplua nyeem
Ntsiav tshuaj: 6 hli round tuag, 8-10knights ntsiav tshuaj
Zaj duab xis txheej: Gastro - soluble zaj duab xis txheej kom txhim kho kev ruaj khov thiab palatability
Kev Tswj Xyuas Zoo:
Cov ntsiab lus sib xyaw: RSD tsawg dua lossis sib npaug ntawm 3% (UV {{1} hplc nrhiav kom pom)
Tus lej sib cais: Ntau dua los yog sib npaug rau 85% hauv 30 feeb (duav txheej txheem, 50 rpm)
Lwm yam tshuaj: Ib leeg impurity tsawg dua los yog sib npaug rau 0.5%, tag nrho cov impurities tsawg dua los yog sib npaug rau 1.0%
2. Npaj sau ntawv:
Cov Khoom Siv Raw Khoom Raw: tsis - steroidal qauv, txom dej solubility
Ib Cheeb Tsam Ntau Lawm: txheeb ze cov av noo tsawg dua los yog sib npaug 40%, noo noo - eam pov thawj kho
Ntim yuav tsum tau: Aluminium ntawv ci tshuab ntim, lub teeb - ntawv pov thawj thiab noo noo-
Vim li cas thiaj xaiv Aastrozole?
Siab xaiv Aromatase inhibitorNrog kev pheej hmoo ntawm cov kev mob tshwm sim
Muaj zog estrogen tswj, txhim khu kev qha nyhuv
Kev thev siab zoothiab muaj kev nyab xeeb rau lub sijhawm ntev - tsis siv
Kev Muaj Peev Xwm Zoo:
GMP -} ua tiav ntau lawm, txhua pobHPLC Purity kuaj (loj dua lossis sib npaug rau 98%)
Thib peb - tog kab ke ceeb toom (COA)suav nrog cov khoom
Microbial txwv kuajTxhawm rau kom muaj kev nyab xeeb
Lub Ntiaj Teb Shipping:
Thawj Ntim Ntim Ntim, noo noo - ntawv pov thawj thiab lub teeb- ntawv pov thawj
Ntiav neeg, tsis muaj logo ntawm lub ntim sab nraud
Kub -} tswj kev thauj mus losTxhawm rau kom muaj kev ruaj khov
Tag
Aastrozole tuaj yeem yogtsim rau hauv kev siv cov tshuaj lim dej siv cov txheej txheem txheemCov. Nws yog tshwj xeeb rauKev kho mob cancer mis, kev tiv thaiv ntawm estrogen -}} kev phiv, thiab cov tshuaj estrogen thaum lub sij hawm steroidCov. Cov koob tshuaj pom zoo yog1 mg / hnub.
Xav tau phiaj xwm npaj phiaj xwm tshwj xeeb?
Peb muab cov kev coj ua kev tshaj lij los pab koj npaj cov khoom kawg kom nyab xeeb thiab zoo!
NEED dab tsi, thov hu raupeb
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Ntawv xov |
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Cim npe nrov: Aastrozole (ArimideX) 99% Hmoov Nplej, Tuam Tshoj areask) 99% Cov Khoom Siv Hmoov Nplej, Chaw muag khoom, Hoobkas

