Dermorphin 5Mg / BUTY CUAM QHIB
Kev Tshawb Nrhiav {{{}}}} grade gradeilized hmoov|Muaj zog {{{- eciod receptor agonist peptide
Amino Acid Seas: H - tyr -}}}}} {}- nh₂
Molecular hnyav: kwv yees li 800 da
Purity: ntau dua los yog sib npaug rau 98% (HPLC)
Cov Lus Qhia Tshwj Xeeb: 5mg / Lub raj mis
Tsos: Dawb khov -} wried hmoov
Kaus: 1ML Cov Dej 1ML Bacteriostatic
Cov teebmeem tseem ceeb
Dermorphin yog aMuaj zog analgesic peptide cais los ntawm daim tawv nqaij ntawm South American Tsob Ntoo Qav QavCov. Vim nwsMuaj kev xaiv thiab muaj zog μ {- opioid receptor agonist cov khoom, nws yog dav siv nyob rau hauvKev Tswj Xyuas Qhov Mob Kev tshawb fawb, neuroscience, thiab opioid receptor chaw muag tshuaj.
✅ Muaj zog analgesic nyhuv:
Muaj kev xaiv siab tau μ {- opioid receptors, nrog ib qho kev ua kom muaj txiaj ntsig 30-40 zaug ntawm morphine
Ntev -} kav cov nyhuv analgesic, ib koob tshuaj tuaj yeem nyob ntev 4-6 teev
✅ Cov Qauv Cov Txheej Txheem Tshwj Xeeb:
Muaj d - amino acid residues (d {{1}- alanine)los tiv thaiv kev tiv thaiv kev ntxhov siab
Txhim Kho Kev Ruaj Ntsegthiab txuas ib nrab - lub neej
✅ Tshawb nrhiav cov ntawv thov zoo:
High receptor xaiv, kev kawm paub tseeb ntawm μ - eciod receptor muaj nuj nqi
Muaj zog analgesic kev ua si, ib qho cuab yeej zoo tagnrho rau kev sim siv lub tshuab kuaj mob
✅ Qhov Zoo:
Haib analgesia, deb dua li ib txwm opioids
Siab heev xaiv, nrog tsawg kev pheej hmoo ntawm cov kev mob tshwm sim
Cov kev siv raws tu qauv
1. Txoj kev hloov kho:
Siv 1ml ntawm cov dej tawgKom maj mam txhaj rau hauv phab ntsa ntawm khov -}} qhuav hmoov lub raj mis
Maj mam yujkom txog thaum yaj tag; tsis txhob tshee tshee los yog vortexing
Cia Tom Qab Rov Kho Dua: Hauv lub tub yees ntawm 2-8℃thiab siv tsis pub dhau 7 hnub
2. Txhaj tshuaj:
Kev txhaj tshuaj: Subcutaneous, entravenous, lossis intrathecal
Txhaj tshuaj txhaj:
Kev Tshawb Fawb Txog Analgesia: 10-50 ug / kg (tsiaj qauv)
Txais Kev Kawm RECTOR: 0.1-1NM (hauv vitro)
Txhaj cev: Txiav txim raws li kev tshawb fawb xav tau
3. Cov ntawv thov kev sim:
Mob Qauv Mob: Mob siab thiab ua mob tsiaj
Kev Tshawb Fawb Dua: {- o o opioid receptor muaj nuj nqi thiab teeb liab transduction kev tshawb fawb
Tshuaj Kho Mob Tshuaj: Kev tshuaj ntsuam thiab ntsuas ntawm cov tshuaj tshiab analgesic
Cov Lus Qhia Cia
1. Kev tsis raws cai:
Kub: {{{- 20℃rau ntev- sijt cia, 2-8℃cia
Vaum: txheeb ze cov av noo tsawg dua los yog sib npaug rau 30%, kev tiv thaiv desiccant
Lub Teeb: Muab tawm ntawm lub teeb, hauv lub raj xim av lossis qhwv hauv txhuas ntawv ci
Hnub tas sij hawm: 24 lub hlis ntawm -20 degree, 12 lub hlis ntawm 2-8 degree
2. Cia Tom Qab Rov Kho Dua:
Siv tam sim ntawd: Rau cov txiaj ntsig zoo tshaj plaws, siv tam sim ntawd tom qab rov kho dua
Khaws rau hauv tub yees: 2-8℃rau tsis pub dhau 7 hnub
Zam kev cia khov: Kev daws teeb meem yuav tsum tsis txhob rov ua khov thiab yaj
3. Thauj cov xwm txheej:
Ultra - Qhov Kub Kub Kub: qhuav thauj khoom (-78 degree)
Ntim Ntim Ntim: Tiv thaiv kev co loj los ntawm kev cuam tshuam peptide qauv
Tus me nyuam sai: Xa tawm hauv 48 teev kom muaj kev ua si
Vim li cas thiaj xaiv dermorphin?
Lub zog μ {- opioid receptor agonistnrog ib qho kev ua kom muaj txiaj ntsig 30-40 zaug ntawm morphine
Cov D - Amino Acid Qauv, txhim kho kev ruaj khov thiab bioavailability
High receptor xaiv, kev kawm paub tseeb ntawm μ - eciod receptor muaj nuj nqi
Kev Muaj Peev Xwm Zoo:
GMP -} ua tiav ntau lawm, txhua pobHPLC Purity kuaj (loj dua lossis sib npaug rau 98%)
Thib peb - tog kab ke ceeb toom (COA)suav nrog cov khoom
Sterile khov khov -}} Kev Siv Kom QhuavTxhawm rau kom tsis muaj endotoxin
Lub Ntiaj Teb Shipping:
Kho Mob Vial Ntim, roj hmab nres foob
Kev Thauj Mus Los QhuavTxhawm rau kom peptide kev ua si
Ntiav neeg, tsis muaj logo ntawm lub ntim sab nraud
Tag
Dermorphin yogIb qho cuab yeej tseem ceeb rau kev tshawb fawb mob thiab Opioid receptor cov kev tshawb fawbCov. Nws yog tshwj xeeb raukawm analgesic kev ua haujlwm, tshawb txog μ -} o o o o opioid receptor muaj nuj nqi, thiab txhim kho cov tshuaj tshiab analgesicCov. Cov koob tshuaj pom zoo yog10-50 ug / kg (hauv tsiaj tsiaj).
Xav tau cov phiaj xwm kev tshawb fawb tshwj xeeb?
Peb muab cov kev coj ua kev tshaj lij pab koj ua koj cov kev tshawb fawb kev nyab xeeb thiab zoo!
Xav taudab tsi, thov hu raupeb
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Cim npe nrov: dermorphin 5mg / vial peptides khov - dermorphin 5mg / vial} qhuav hmoov tuam ntxhab, lwm tus neeg, Hoobkas

